SCHEMBL2567253

SCHEMBL2567253

Cc1cc(C)c(S(=O)(=O)N2Cc3ccccc3CC2COCC(=O)NCc2cccc(N3CCOCC3)c2)c(C)c1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP8 P22894 2/20 0.40
MMP3 P08254 1/20 0.40
EPHX2 P34913 3/20 0.39
KMT2A Q03164 3/20 0.39
LMNA P02545 2/20 0.39
MEN1 O00255 1/20 0.39
TSHR P16473 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PKM P14618 1/20 0.38
KLKB1 P03952 1/20 0.37
KLK1 P06870 1/20 0.37
POLB P06746 1/20 0.36
MAPT P10636 2/20 0.36
TRPA1 O75762 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2566667 0.93 EPHX2 (0.40) EPHX2KMT2ALMNAPKMMAPT
SCHEMBL2567533 0.81 EPHX2 (0.42) EPHX2LMNANPSR1PKM
SCHEMBL2568675 0.80 EPHX2 (0.41) EPHX2KMT2ALMNAMEN1TSHR
SCHEMBL2564993 0.80 MEN1 (0.41) KMT2AMEN1POLBMAPT
SCHEMBL5127128 0.77 EPHX2 (0.43) EPHX2KMT2AMEN1POLBMAPT
SCHEMBL2565172 0.76 MMP8 (0.49) MMP8MMP3LMNAPOLBMAPT
SCHEMBL2564561 0.73 MEN1 (0.45) KMT2AMEN1TRPA1
SCHEMBL2569446 0.73 GFER (0.42) KMT2AMEN1TRPA1
SCHEMBL2570767 0.72 MAPT (0.42) MMP8MMP3KMT2ALMNAMEN1
SCHEMBL2565909 0.72 POLB (0.47) TSHRPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2383267-A1 Substituted sulfonamide derivatives Grünenthal GmbH (DE) 2011-11-02 EP claimed
US-20100317644-A1 Substituted Sulfonamide Compounds GRUENENTHAL GMBH (DE) 2010-12-16 US claimed
US-20080153843-A1 SUBSTITUTED SULFONAMIDE COMPOUNDS GRUENENTHAL GMBH (DE) 2008-06-26 US claimed
US-8435978-B2 Substituted sulfonamide compounds GRUENENTHAL GMBH (DE) 2013-05-07 US disclosed
EP-2383267-A1 Substituted sulfonamide derivatives Grünenthal GmbH (DE) 2011-11-02 EP disclosed
US-20100324009-A1 Substituted Sulfonamide Compounds GRUENENTHAL GMBH (DE) 2010-12-23 US disclosed
US-20100317644-A1 Substituted Sulfonamide Compounds GRUENENTHAL GMBH (DE) 2010-12-16 US disclosed
US-20080153843-A1 SUBSTITUTED SULFONAMIDE COMPOUNDS GRUENENTHAL GMBH (DE) 2008-06-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100317644-A1 Substituted Sulfonamide Compounds SULT2A1, STS, SULT1A1 MMP8 2055/4885MMP3 3494/4885EPHX2 2401/4885
US-20100324009-A1 Substituted Sulfonamide Compounds SULT2A1, STS, SULT1A1 MMP8 2055/4885MMP3 3494/4885EPHX2 2401/4885
US-20080153843-A1 SUBSTITUTED SULFONAMIDE COMPOUNDS SULT2A1, STS, SULT1A1 MMP8 2055/4885MMP3 3494/4885EPHX2 2401/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.