SCHEMBL25692091

SCHEMBL25692091

CSN(C)c1ccccc1Nc1nc(Cl)ncc1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ULK1 O75385 4/20 0.44
PTK2 Q05397 5/20 0.41
MAPK3 P27361 4/20 0.39
CDK1 P06493 1/20 0.39
CDK4 P11802 1/20 0.39
CDK2 P24941 1/20 0.39
CDC7 O00311 1/20 0.39
ROCK2 O75116 1/20 0.39
MAP4K4 O95819 1/20 0.39
PIM1 P11309 1/20 0.39
PRKACA P17612 1/20 0.39
CDK7 P50613 1/20 0.39
CDK9 P50750 1/20 0.39
HIPK2 Q9H2X6 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.39
KDR P35968 2/20 0.38
JAK2 O60674 1/20 0.38
NTRK1 P04629 1/20 0.38
TYK2 P29597 1/20 0.38
JAK3 P52333 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25234927 0.83 PTK2 (0.49) PTK2PTK2B
SCHEMBL24716006 0.83 ULK1 (0.48) ULK1PTK2MAPK3CDK1CDK4
SCHEMBL25056242 0.81 IGF1R (0.48) IGF1RLRRK2
SCHEMBL17102732 0.79 PTK2 (0.45) ULK1PTK2MAPK3CDC7ROCK2
SCHEMBL12813038 0.77 CDC7 (0.52) ULK1PTK2MAPK3CDC7ROCK2
SCHEMBL28295859 0.77 ULK1 (0.47) ULK1PTK2MAPK3CDK1CDK4
SCHEMBL25692191 0.76 GSK3A (0.69) PTK2MAPK3CDC7ROCK2MAP4K4
SCHEMBL24715923 0.76 ULK1 (0.44) ULK1PTK2MAPK3CDK1CDK4
SCHEMBL28969607 0.76 ULK1 (0.52) ULK1PTK2MAPK3CDK1CDK4
SCHEMBL19831480 0.75 CDC7 (0.50) ULK1PTK2MAPK3CDC7ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023121251-A1 EGFR AND HDAC DUAL INHIBITOR COMPOUNDS AND MEDICAL USE THEREOF 한국원자력의학원 2023-06-29 WO disclosed