SCHEMBL25713579

SCHEMBL25713579

C=CC(=O)N1CCn2c(nc(C)c2C)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.38
ACHE P22303 3/20 0.35
HTT P42858 1/20 0.33
TSHR P16473 1/20 0.33
BTK Q06187 3/20 0.33
RYR2 Q92736 1/20 0.33
JAK3 P52333 3/20 0.31
P2RX7 Q99572 1/20 0.31
TACR3 P29371 2/20 0.31
TET3 O43151 1/20 0.31
KMT2A Q03164 1/20 0.31
FBXL19 Q6PCT2 1/20 0.31
CXXC5 Q7LFL8 1/20 0.31
TET1 Q8NFU7 1/20 0.31
KDM2B Q8NHM5 1/20 0.31
CXXC4 Q9H2H0 1/20 0.31
KDM2A Q9Y2K7 1/20 0.31
EGFR P00533 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25976628 0.72 NOTUM (0.40) MAPK1ACHEBTKRYR2JAK3
SCHEMBL25976627 0.71 P2RX7 (0.53) MAPK1ACHEBTKRYR2JAK3
SCHEMBL31065977 0.68 TSHR (0.38) HTTTSHRP2RX7TACR3CYP1A2
SCHEMBL19042592 0.67 DPP4 (0.51)
SCHEMBL25976602 0.66 MAPK1 (0.50) MAPK1ACHEBTKRYR2EGFR
SCHEMBL25976625 0.66 MAPK1 (0.38) MAPK1ACHEBTKRYR2TET3
SCHEMBL24639555 0.66 POLB (0.38) MAPK1TSHRBTKJAK3P2RX7
SCHEMBL12764449 0.64 TET3 (0.47) MAPK1ACHETSHRJAK3TET3
SCHEMBL167151 0.64 TET3 (0.47) MAPK1ACHETSHRJAK3TET3
SCHEMBL20547259 0.64 TET3 (0.47) MAPK1ACHETSHRJAK3TET3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023104035-A1 SUBSTITUTED MONOCYCLIC OR BICYCLIC HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 英矽智能科技(上海)有限公司 2023-06-15 WO disclosed