SCHEMBL257187

SCHEMBL257187

CC(Cc1ccccc1)[C@H](O)CNCc1cccc(CC(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 10/20 0.49
BCHE P06276 8/20 0.49
TRPA1 O75762 1/20 0.47
CTSD P07339 1/20 0.41
BACE2 Q9Y5Z0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5216600 0.85 BACE1 (0.49) BACE1BCHE
SCHEMBL256560 0.78 BCHE (0.46) BACE1BCHE
SCHEMBL14201586 0.76 BACE1 (0.54) BACE1CTSD
SCHEMBL7909784 0.74 TRPA1 (0.61) BCHETRPA1
SCHEMBL19567292 0.73 CYP1A2 (0.41)
SCHEMBL20781990 0.71 SLC2A1 (0.47)
SCHEMBL13073581 0.71 BCHE (0.48) BACE1BCHE
SCHEMBL4043821 0.71 BACE1 (0.48) BACE1BCHE
SCHEMBL8276492 0.71 BACE1 (0.62) BACE1BCHECTSDBACE2
SCHEMBL3455222 0.71 BACE1 (0.62) BACE1BCHECTSDBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012028563-A1 BACE INHIBITORS FOR USE IN THE TREATMENT OF DIABETES F. HOFFMANN-LA ROCHE AG (CH) 2012-03-08 WO disclosed