SCHEMBL2572035

SCHEMBL2572035

O=C(O)N1CC(Cn2cccn2)C1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.37
FDPS P14324 1/20 0.37
TSHR P16473 2/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
KMT2A Q03164 2/20 0.34
GFER P55789 2/20 0.33
ENPP2 Q13822 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
MEN1 O00255 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
KDM5A P29375 1/20 0.31
KDM2B Q8NHM5 1/20 0.31
KDM4C Q9H3R0 1/20 0.31
KDM5B Q9UGL1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25412012 0.88 ENPP2 (0.38) HTTFDPSTSHRKMT2AGFER
SCHEMBL20297422 0.85 GFER (0.41) KMT2AGFER
SCHEMBL9935087 0.84 HTT (0.35) HTTFDPSTSHRHDAC1HDAC6
SCHEMBL9935089 0.84 HTT (0.35) HTTFDPSTSHRHDAC1HDAC6
SCHEMBL4290754 0.75 CA1 (0.34) HTTFDPSGFER
SCHEMBL5141170 0.74
SCHEMBL30515619 0.71 GPR119 (0.45)
SCHEMBL14857835 0.71 CYP2B6 (0.44) FDPSTSHRKMT2A
SCHEMBL6155217 0.71 CYP2B6 (0.40) FDPSTSHRKMT2AHRH3
SCHEMBL17229398 0.70 NOS1 (0.39) FDPSTSHRKMT2AENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2384328-A1 6,7,8,9-TETRAHYDRO-5H-1,4,7,10A-TETRAAZA-CYCLOHEPT[F]INDENE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR PREPARING THEM Boehringer Ingelheim International GmbH (DE) 2011-11-09 EP disclosed
WO-2010060952-A1 6,7,8,9-TETRAHYDRO-5H-1,4,7,10A-TETRAAZA-CYCLOHEPT[F]INDENE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-06-03 WO disclosed