SCHEMBL2573370

SCHEMBL2573370

O=C(O)N1CCCCCC1(F)F

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ALDH1A1 P00352 2/20 0.31
HSD11B1 P28845 1/20 0.31
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20919200 0.98 MEN1 (0.31) MEN1KMT2A
SCHEMBL23795144 0.91
SCHEMBL4027926 0.82 ALDH1A1 (0.33) ALDH1A1
SCHEMBL23795158 0.81
SCHEMBL3430843 0.78 MEN1 (0.30) MEN1KMT2A
SCHEMBL28743535 0.73 CYP2C19 (0.32) MEN1KMT2AHSD11B1CYP2C19
SCHEMBL25365469 0.73 MEN1 (0.32) MEN1KMT2A
SCHEMBL31691566 0.73 MEN1 (0.32) MEN1KMT2A
SCHEMBL28236926 0.73 MEN1 (0.32) MEN1KMT2A
SCHEMBL14970353 0.71 EPHX2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2384328-A1 6,7,8,9-TETRAHYDRO-5H-1,4,7,10A-TETRAAZA-CYCLOHEPT[F]INDENE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR PREPARING THEM Boehringer Ingelheim International GmbH (DE) 2011-11-09 EP disclosed
WO-2010060952-A1 6,7,8,9-TETRAHYDRO-5H-1,4,7,10A-TETRAAZA-CYCLOHEPT[F]INDENE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-06-03 WO disclosed