SCHEMBL257346

SCHEMBL257346

Bc1ccc(C(=O)O)c(C)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRB P28702 2/20 0.49
RXRA P19793 1/20 0.47
CYP1A2 P05177 1/20 0.44
HAAO P46952 1/20 0.44
ALDH1A1 P00352 3/20 0.43
MYC P01106 1/20 0.43
RARB P10826 1/20 0.42
GABRP O00591 2/20 0.42
GABRD O14764 2/20 0.42
GABRA1 P14867 2/20 0.42
GABRB1 P18505 2/20 0.42
GABRG2 P18507 2/20 0.42
GABRB3 P28472 2/20 0.42
GABRA5 P31644 2/20 0.42
GABRA3 P34903 2/20 0.42
GABRA2 P47869 2/20 0.42
GABRB2 P47870 2/20 0.42
GABRA4 P48169 2/20 0.42
GABRE P78334 2/20 0.42
GABRA6 Q16445 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14366361 0.84 MCL1 (0.43) CYP1A2HAAOALDH1A1MYCGABRP
SCHEMBL13652578 0.81 ALDH1A1 (0.48) CYP1A2HAAOALDH1A1KDM4EHSD17B10
SCHEMBL30679777 0.79 CSNK2A1 (0.59) RXRBRXRAALDH1A1KDM4ECSNK2A1
SCHEMBL29399874 0.79 MYC (0.58) RXRBRXRACYP1A2ALDH1A1MYC
SCHEMBL44342 0.79 MYC (0.58) RXRBRXRACYP1A2ALDH1A1MYC
SCHEMBL29771992 0.79 RXRB (0.70) RXRBRXRACYP1A2RARBKDM4E
SCHEMBL1498034 0.79 RXRB (0.70) RXRBRXRACYP1A2RARBKDM4E
SCHEMBL107259 0.79 CSNK2A1 (0.59) RXRBRXRAALDH1A1KDM4ECSNK2A1
SCHEMBL6915656 0.77 CSNK2A1 (0.57) RXRBRXRAALDH1A1KDM4ECSNK2A1
Water SCHEMBL3832510 0.77 MYC (0.56) RXRBRXRACYP1A2ALDH1A1MYC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108368083-B Heteroaryl compounds and their use as therapeutic agents 东亚首希控股股份有限公司 2022-02-01 CN disclosed
WO-2012029942-A1 CYCLIC AMIDE DERIVATIVE 大日本住友製薬株式会社 (JP) 2012-03-08 WO disclosed
WO-2009126863-A2 PYRIDYL INHIBITORS OF HEDGEHOG SIGNALLING GENENTECH, INC. (US) 2009-10-15 WO disclosed