SCHEMBL257382

SCHEMBL257382

Cc1ccc(-c2c(C)nn3c(-c4ccc(F)cc4)cc(Cl)nc23)cc1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.53
MAPT P10636 11/20 0.51
MAPK1 P28482 1/20 0.46
THRB P10828 1/20 0.46
KMT2A Q03164 3/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HTT P42858 1/20 0.45
POLB P06746 1/20 0.45
HPGD P15428 1/20 0.45
NPC1 O15118 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15042157 0.88 TP53 (0.67) TP53MAPTMAPK1KMT2AMEN1
SCHEMBL10072008 0.88 TP53 (0.52) TP53MAPTMAPK1THRBKMT2A
SCHEMBL257503 0.85 ALDH1A1 (0.50) TP53MAPTTHRBKMT2AALDH1A1
SCHEMBL13516316 0.84 MAPT (0.66) TP53MAPTTHRBKMT2AMEN1
SCHEMBL257542 0.84 TP53 (0.55) TP53MAPTMAPK1KMT2AMEN1
SCHEMBL256955 0.82 ALDH1A1 (0.40) TP53MAPTTHRBALDH1A1HPGD
SCHEMBL257314 0.82 TP53 (0.41) TP53MAPTMAPK1THRBKMT2A
SCHEMBL256953 0.81 MAPT (0.41) TP53MAPTMAPK1THRBKMT2A
SCHEMBL15020632 0.81 TP53 (0.79) TP53MAPTMAPK1KMT2AMEN1
SCHEMBL257701 0.80 TP53 (0.49) TP53MAPTMAPK1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8975264-B2 Compound acting as a cannabinoid receptor-1 inhibitor AMOREPACIFIC CORPORATION (KR) 2015-03-10 US disclosed
US-8975264-B2 Compound acting as a cannabinoid receptor-1 inhibitor AMOREPACIFIC CORPORATION (KR) 2015-03-10 US disclosed
US-8975264-B2 Compound acting as a cannabinoid receptor-1 inhibitor AMOREPACIFIC CORPORATION (KR) 2015-03-10 US disclosed
US-20130158025-A1 NOVEL COMPOUND ACTING AS A CANNABINOID RECEPTOR-1 INHIBITOR AMOREPACIFIC CORPORATION (KR) 2013-06-20 US disclosed
US-20130158025-A1 NOVEL COMPOUND ACTING AS A CANNABINOID RECEPTOR-1 INHIBITOR AMOREPACIFIC CORPORATION (KR) 2013-06-20 US disclosed
US-20130158025-A1 NOVEL COMPOUND ACTING AS A CANNABINOID RECEPTOR-1 INHIBITOR AMOREPACIFIC CORPORATION (KR) 2013-06-20 US disclosed
WO-2012030170-A2 NOVEL COMPOUND ACTING AS A CANNABINOID RECEPTOR-1 INHIBITOR (주)아모레퍼시픽 (KR) 2012-03-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130158025-A1 NOVEL COMPOUND ACTING AS A CANNABINOID RECEPTOR-1 INHIBITOR CNR1, CNR2, GPR18 TP53 4550/4885MAPT 2617/4885MAPK1 519/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.