SCHEMBL2574754

SCHEMBL2574754

CC(C)CNc1cc(C2Nc3ccc(C(=O)O)cc3CC2(C)C)ccc1F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 1/20 0.35
HCAR2 Q8TDS4 1/20 0.35
PRKAG1 P54619 2/20 0.34
PRKAA1 Q13131 2/20 0.34
PRKAB1 Q9Y478 2/20 0.34
PRKAB2 O43741 1/20 0.34
PRKAA2 P54646 1/20 0.34
PRKAG3 Q9UGI9 1/20 0.34
PRKAG2 Q9UGJ0 1/20 0.34
CREBBP Q92793 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32
APOBEC3A P31941 1/20 0.32
APOBEC3G Q9HC16 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
RXRA P19793 1/20 0.31
HNF4A P41235 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2589366 0.91 SMN1; SMN2 (0.38) MEN1KMT2AALDH1A1GAAL3MBTL1
SCHEMBL2565976 0.89 CASR (0.35) HCAR3HCAR2CREBBPMEN1KMT2A
SCHEMBL2529499 0.86 CYP26A1 (0.36) PRKAG1PRKAA1PRKAB1PRKAB2PRKAA2
SCHEMBL2574265 0.85 HCAR3 (0.38) HCAR3HCAR2MEN1KMT2AALDH1A1
SCHEMBL2567515 0.83 KDM4E (0.37) HCAR3PRKAG1PRKAA1PRKAB1PRKAB2
SCHEMBL2529993 0.82 TSHR (0.39) PRKAG1PRKAA1PRKAB1PRKAB2PRKAA2
SCHEMBL2533068 0.82 PPARG (0.46) HCAR3CREBBPMEN1KMT2A
SCHEMBL2574406 0.82 ITGB3 (0.41) ALDH1A1
SCHEMBL2532031 0.81 PPARG (0.38) CREBBPKMT2AGAALMNA
SCHEMBL2531335 0.81 KMT2A (0.41) PRKAG1PRKAA1PRKAB1PRKAB2PRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2558449-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2013-02-20 EP disclosed
WO-2011128251-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-10-20 WO disclosed