SCHEMBL2589366

SCHEMBL2589366

COC(=O)c1ccc2c(c1)CC(C)(C)C(c1ccc(F)c(NCC(C)C)c1)N2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
MEN1 O00255 5/20 0.36
KMT2A Q03164 5/20 0.36
ALDH1A1 P00352 3/20 0.36
AR P10275 1/20 0.35
MAPT P10636 6/20 0.32
KDM4E B2RXH2 4/20 0.32
MAPK1 P28482 2/20 0.32
CRBN Q96SW2 1/20 0.32
GAA P10253 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HTT P42858 2/20 0.32
GLA P06280 1/20 0.32
CASP1 P29466 1/20 0.32
KLK7 P49862 1/20 0.32
CASP7 P55210 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HPGD P15428 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2574754 0.91 HCAR3 (0.35) MEN1KMT2AALDH1A1GAAL3MBTL1
SCHEMBL2576665 0.89 ALDH1A1 (0.39) SMN1; SMN2RAB9ANPC1MEN1KMT2A
SCHEMBL2532967 0.86 ALDH1A1 (0.43) SMN1; SMN2RAB9ANPC1MEN1KMT2A
SCHEMBL2568952 0.86 CRBN (0.39) SMN1; SMN2RAB9ANPC1MEN1KMT2A
SCHEMBL2536690 0.83 ALDH1A1 (0.46) SMN1; SMN2RAB9ANPC1MEN1KMT2A
SCHEMBL2578929 0.82 VNN1 (0.38) SMN1; SMN2RAB9ANPC1MEN1KMT2A
SCHEMBL2535519 0.82 MAPK14 (0.47) RAB9ANPC1MEN1KMT2AKDM4E
SCHEMBL2527678 0.82 GRM4 (0.39) SMN1; SMN2RAB9ANPC1MEN1KMT2A
SCHEMBL2527848 0.81 ALDH1A1 (0.42) SMN1; SMN2RAB9ANPC1MEN1KMT2A
SCHEMBL2534017 0.81 ALDH1A1 (0.42) SMN1; SMN2RAB9ANPC1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2558449-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2013-02-20 EP disclosed
WO-2011128251-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-10-20 WO disclosed