SCHEMBL25754850

SCHEMBL25754850

Cc1ccc2c(c1)CCN2S(=O)(=O)c1cccc(N)c1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
ATM Q13315 1/20 0.55
DRD3 P35462 5/20 0.53
HTR6 P50406 4/20 0.53
TP53 P04637 2/20 0.52
CYP11B1 P15538 2/20 0.49
CYP11B2 P19099 2/20 0.49
HRH3 Q9Y5N1 2/20 0.49
DRD2 P14416 2/20 0.49
TNF P01375 1/20 0.48
NOD2 Q9HC29 1/20 0.48
NOD1 Q9Y239 1/20 0.48
AKR1C3 P42330 1/20 0.48
AKR1C1 Q04828 1/20 0.48
MAPT P10636 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5475972 0.84 AKR1C3 (0.66) MEN1KMT2AATMTP53AKR1C3
SCHEMBL5460641 0.81 KMT2A (0.61) MEN1KMT2AATMDRD3HTR6
SCHEMBL25754772 0.81 KMT2A (0.55) MEN1KMT2AATMDRD3HTR6
SCHEMBL5479450 0.80 TP53 (0.53) MEN1KMT2AATMTP53MAPT
SCHEMBL25754845 0.79 PKM (0.52) MEN1KMT2AATMHTR6MAPT
SCHEMBL2693546 0.79 MEN1 (0.85) MEN1KMT2AATMAKR1C3AKR1C1
SCHEMBL23847014 0.78 KMT2A (0.59) MEN1KMT2AATMTP53CYP11B1
SCHEMBL4115320 0.76 KMT2A (0.72) MEN1KMT2AATMTP53AKR1C3
SCHEMBL5472746 0.75 KMT2A (0.67) MEN1KMT2AATMTP53AKR1C3
SCHEMBL5474194 0.74 KMT2A (0.65) MEN1KMT2AATMTP53AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2023-06-08 US disclosed
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2023-06-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF TRAP1, PINK1, TP53BP1 MEN1 3902/4885KMT2A 4864/4885ATM 652/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.