SCHEMBL2575501

SCHEMBL2575501

CC(C)(C)OC(=O)N[C@@](C)(CCC(=O)c1ccc(F)c(F)c1)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA1 P02708 1/20 0.38
CHRNG P07510 1/20 0.38
CHRNB1 P11230 1/20 0.38
CHRNB2 P17787 1/20 0.38
SLC6A2 P23975 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
SLC6A3 Q01959 1/20 0.38
CHRND Q07001 1/20 0.38
TRPA1 O75762 1/20 0.36
ALDH1A1 P00352 3/20 0.36
AAK1 Q2M2I8 2/20 0.36
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
NAALAD2 Q9Y3Q0 1/20 0.35
RAB9A P51151 3/20 0.35
MAPT P10636 2/20 0.35
HPGD P15428 2/20 0.35
NPC1 O15118 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2581131 0.93 DRD2 (0.37) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL22039571 0.86 AAK1 (0.40) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL23878364 0.86 LMNA (0.46) ALDH1A1NAALAD2RAB9ANPC1MEN1
SCHEMBL2581151 0.85 CHRNA1 (0.36) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL4330484 0.81 AAK1 (0.34) TRPA1AAK1CES2CES1NAALAD2
SCHEMBL1093048 0.78 NOX1 (0.45) ALDH1A1RAB9AMAPTHPGDNPC1
SCHEMBL310957 0.78 MAOB (0.51) ALDH1A1RAB9ANPC1LMNACTSS
SCHEMBL4092905 0.78 PPARA (0.49) TRPA1ALDH1A1MAPTCTSSCTSK
SCHEMBL4514578 0.78 PPARA (0.49) TRPA1ALDH1A1MAPTCTSSCTSK
SCHEMBL4092912 0.78 PPARA (0.49) TRPA1ALDH1A1MAPTCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048878-B2 Two cyclic cinnamide compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2011-11-01 US disclosed