SCHEMBL2581151

SCHEMBL2581151

CC[C@@](CCC(=O)c1ccc(F)c(F)c1)(NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA1 P02708 1/20 0.36
CHRNG P07510 1/20 0.36
CHRNB1 P11230 1/20 0.36
CHRNB2 P17787 1/20 0.36
SLC6A2 P23975 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
SLC6A3 Q01959 1/20 0.36
CHRND Q07001 1/20 0.36
ALDH1A1 P00352 5/20 0.36
MAPT P10636 5/20 0.36
RAB9A P51151 3/20 0.36
HPGD P15428 3/20 0.36
NPC1 O15118 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TRPA1 O75762 1/20 0.35
THRA P10827 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2584672 0.89 AAK1 (0.34) ALDH1A1MAPTRAB9AHPGDTRPA1
SCHEMBL2587439 0.86 CTSS (0.41) MAPTRAB9AHPGDNPC1MEN1
SCHEMBL2575528 0.85 ALDH1A1 (0.47) ALDH1A1MAPTHPGDMEN1KMT2A
SCHEMBL2585429 0.85 CTSS (0.33) SLC6A3AAK1GABRB1GABRB2
SCHEMBL2575501 0.85 CHRNA1 (0.38) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL2588069 0.84 AAK1 (0.34) AAK1
SCHEMBL22039571 0.83 AAK1 (0.40) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL2583802 0.83 ERCC5 (0.42) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL2587766 0.83 CTSS (0.35) ALDH1A1MAPTHPGDMEN1KMT2A
SCHEMBL2584542 0.82 CES2 (0.33) ALDH1A1MAPTHPGDAAK1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048878-B2 Two cyclic cinnamide compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2011-11-01 US disclosed