SCHEMBL25757652

SCHEMBL25757652

O=C1NCc2c1ccc1nc[nH]c21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 2/20 0.41
DYRK1A Q13627 2/20 0.41
CLK4 Q9HAZ1 2/20 0.41
PIM1 P11309 2/20 0.41
CSNK1A1 P48729 1/20 0.41
ROCK1 Q13464 1/20 0.41
LRRK2 Q5S007 1/20 0.41
DYRK1B Q9Y463 1/20 0.41
MKNK1 Q9BUB5 1/20 0.40
KDM4A O75164 1/20 0.37
KDM4B O94953 1/20 0.37
KDM5C P41229 1/20 0.37
KDM4C Q9H3R0 1/20 0.37
KDM5B Q9UGL1 1/20 0.37
KDM3A Q9Y4C1 1/20 0.37
LTK P29376 1/20 0.36
MST1R Q04912 1/20 0.36
CYP17A1 P05093 1/20 0.36
CYP3A4 P08684 1/20 0.36
CA12 O43570 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31451620 1.00 CDK5 (0.41) CDK5DYRK1ACLK4PIM1CSNK1A1
SCHEMBL6807733 0.73 DYRK1A (0.41) CDK5DYRK1ACLK4PIM1CSNK1A1
SCHEMBL11663189 0.69 PARP1 (0.42) PIM1CA12CA9IP6K1IP6K3
SCHEMBL16335317 0.69 DYRK1A (0.40) CDK5DYRK1ACLK4PIM1CSNK1A1
SCHEMBL599458 0.69 DYRK1A (0.42) CDK5DYRK1ACLK4PIM1CSNK1A1
SCHEMBL1374558 0.69 PRKCI (0.44) DYRK1APIM1CYP3A4CA12CA9
SCHEMBL2070779 0.67 NEK2 (0.36) CDK5PIM1KDM4AKDM4BKDM5C
SCHEMBL24466337 0.65 CDK5 (0.46) CDK5DYRK1ACLK4PIM1CSNK1A1
SCHEMBL15566157 0.65 CLK4 (0.46) CDK5DYRK1ACLK4PIM1CSNK1A1
SCHEMBL31264207 0.65 CDK5 (0.46) CDK5DYRK1ACLK4PIM1CSNK1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023098880-A1 FUSED RING DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 上海翰森生物医药科技有限公司 2023-06-08 WO disclosed