SCHEMBL25768628

SCHEMBL25768628

Cc1cc2cc(Oc3c(Cl)cc(-n4nc(C#N)c(=O)[nH]c4=O)cc3Cl)ccc2nc1Cl

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
THRB P10828 19/20 0.53
THRA P10827 16/20 0.53
CYP2C9 P11712 2/20 0.53
CYP2C8 P10632 1/20 0.53
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
OPRK1 P41145 1/20 0.37
HTT P42858 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
UGT1A1 P22309 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.37
SLCO1B1 Q9Y6L6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30460687 1.00 THRB (0.53) THRBTHRACYP2C9CYP2C8NPC1
SCHEMBL31300946 0.89 THRB (0.49) THRBTHRACYP2C9CYP2C8
SCHEMBL25768629 0.89 THRB (0.49) THRBTHRACYP2C9CYP2C8
SCHEMBL23042578 0.88 THRA (0.54) THRBTHRACYP2C9CYP2C8NPC1
SCHEMBL25873840 0.87 THRB (0.53) THRBTHRACYP2C9CYP2C8NPC1
SCHEMBL29612524 0.87 THRB (0.53) THRBTHRACYP2C9CYP2C8NPC1
SCHEMBL22633008 0.86 THRB (0.54) THRBTHRACYP2C9CYP2C8NPC1
SCHEMBL25247755 0.86 THRB (0.51) THRBTHRACYP2C9CYP2C8UGT1A1
SCHEMBL30460689 0.86 THRB (0.51) THRBTHRACYP2C9CYP2C8UGT1A1
SCHEMBL30460733 0.85 THRA (0.52) THRBTHRACYP2C9CYP2C8NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125716-A1 CLASS OF QUINOLINE COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND USE THEREOF 中国科学院上海药物研究所 2023-07-06 WO disclosed
CN-116354934-A Quinoline compound, preparation method, pharmaceutical composition and application thereof 中国科学院上海药物研究所 2023-06-30 CN disclosed