SCHEMBL25768630

SCHEMBL25768630

Cc1cc(-c2ccccc2)nc2ccc(Oc3c(F)cc(-n4nc(C#N)c(=O)[nH]c4=O)cc3F)cc12

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
THRA P10827 13/20 0.38
THRB P10828 13/20 0.38
CYP2C8 P10632 1/20 0.38
CYP2C9 P11712 1/20 0.38
DHODH Q02127 1/20 0.35
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
F10 P00742 1/20 0.33
MET P08581 1/20 0.33
EGLN2 Q96KS0 1/20 0.32
EGLN1 Q9GZT9 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
PLA2G2A P14555 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30460706 1.00 THRA (0.38) THRATHRBCYP2C8CYP2C9DHODH
SCHEMBL31301011 0.93 THRB (0.39) THRATHRBCYP2C8CYP2C9DHODH
SCHEMBL30460702 0.90 THRB (0.49) THRATHRBCYP2C8CYP2C9SMN1; SMN2
SCHEMBL25291901 0.90 THRB (0.49) THRATHRBCYP2C8CYP2C9SMN1; SMN2
SCHEMBL30460745 0.89 THRB (0.37) THRATHRBCYP2C8CYP2C9DHODH
SCHEMBL25769194 0.87 DHODH (0.36) THRATHRBCYP2C9DHODHKDM4E
SCHEMBL30511685 0.87 DHODH (0.36) THRATHRBCYP2C9DHODHKDM4E
SCHEMBL31300999 0.87 THRB (0.44) THRATHRBCYP2C8CYP2C9MEN1
SCHEMBL25768632 0.87 THRB (0.44) THRATHRBCYP2C8CYP2C9MEN1
SCHEMBL30460729 0.86 THRA (0.48) THRATHRBCYP2C8CYP2C9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125716-A1 CLASS OF QUINOLINE COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND USE THEREOF 中国科学院上海药物研究所 2023-07-06 WO disclosed
CN-116354934-A Quinoline compound, preparation method, pharmaceutical composition and application thereof 中国科学院上海药物研究所 2023-06-30 CN disclosed