SCHEMBL257987

SCHEMBL257987

Cc1ccc(Oc2cccc(C(=O)OC(C)C)c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.49
RAB9A P51151 4/20 0.49
SMN1; SMN2 Q16637 4/20 0.49
HTT P42858 2/20 0.49
MAPT P10636 1/20 0.49
TNKS O95271 1/20 0.49
PARP15 Q460N3 1/20 0.49
PARP14 Q460N5 1/20 0.49
PARP10 Q53GL7 1/20 0.49
TNKS2 Q9H2K2 1/20 0.49
PARP2 Q9UGN5 1/20 0.49
AKR1C3 P42330 1/20 0.49
GCK P35557 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11253833 0.89 AKR1C3 (0.62) NPC1RAB9ASMN1; SMN2HTTMAPT
SCHEMBL12260854 0.87 HDAC8 (0.50) NPC1RAB9ASMN1; SMN2HTTMAPT
SCHEMBL257629 0.85 CA1 (0.49) NPC1RAB9ASMN1; SMN2HTTMAPT
SCHEMBL14217726 0.83 L3MBTL1 (0.56) NPC1RAB9ASMN1; SMN2TNKSPARP15
SCHEMBL8737053 0.81 MEN1 (0.60) NPC1RAB9ASMN1; SMN2MAPTTNKS
SCHEMBL8736479 0.80 MAOB (0.63) NPC1RAB9ASMN1; SMN2HTTMAPT
SCHEMBL25910311 0.80 MAOB (0.63) NPC1RAB9ASMN1; SMN2HTTMAPT
SCHEMBL2867826 0.80 AKR1C3 (0.77) NPC1RAB9AHTTTNKSPARP15
SCHEMBL8459413 0.80 CES2 (0.62) NPC1RAB9ASMN1; SMN2HTTMAPT
SCHEMBL6057062 0.79 RAB9A (0.58) NPC1RAB9ASMN1; SMN2HTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2404607-A1 Boronic acids and esters as inhibitors of fatty acid amide hydrolase Infinity Pharmaceuticals, Inc. (US) 2012-01-11 EP disclosed
EP-2399585-A1 Boronic acids and esters as inhibitors of fatty acid amide hydrolase Infinity Pharmaceuticals, Inc. (US) 2011-12-28 EP disclosed
EP-2073816-B1 BORONIC ACIDS AND ESTERS AS INHIBITORS OF FATTY ACID AMIDE HYDROLASE INFINITY PHARMACEUTICALS INC (US) 2011-09-14 EP disclosed