SCHEMBL25804261

SCHEMBL25804261

COc1ccc(CNc2nccc3c2c(C)nn3C(C)C)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.48
CDK1 P06493 3/20 0.47
CCNB2 O95067 2/20 0.47
CCNB1 P14635 2/20 0.47
CCNB3 Q8WWL7 2/20 0.47
TDP1 Q9NUW8 1/20 0.46
PDE1A P54750 2/20 0.45
PDE1B Q01064 2/20 0.45
PDE1C Q14123 2/20 0.45
NPC1 O15118 1/20 0.44
CACNA2D1 P54289 1/20 0.43
KDM4E B2RXH2 1/20 0.42
CHRM4 P08173 1/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
CDK5 Q00535 1/20 0.42
CDK5R1 Q15078 1/20 0.42
PDE5A O76074 1/20 0.42
PDE6C P51160 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30566240 0.87 CDK1 (0.49) THRBCDK1CCNB2CCNB1CCNB3
SCHEMBL25283284 0.87 CDK1 (0.49) THRBCDK1CCNB2CCNB1CCNB3
SCHEMBL25706604 0.86 THRB (0.50) THRBCDK1CCNB2CCNB1CCNB3
SCHEMBL30577105 0.76 PDE1A (0.60) CDK1CCNB2CCNB1CCNB3PDE1A
SCHEMBL25243808 0.75 CDK1 (0.46) THRBCDK1CCNB2CCNB1CCNB3
SCHEMBL30566199 0.75 CDK1 (0.46) THRBCDK1CCNB2CCNB1CCNB3
SCHEMBL25804253 0.73 THRB (0.52) THRBCDK1CCNB2CCNB1CCNB3
SCHEMBL25273214 0.73 CDK1 (0.46) THRBCDK1CCNB2CCNB1CCNB3
SCHEMBL30446331 0.73 CDK1 (0.46) THRBCDK1CCNB2CCNB1CCNB3
SCHEMBL22581153 0.72 CYP1A2 (0.46) TDP1NPC1LMNATP53CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023115150-A1 BIFUNCTIONAL ARYLSULPHONAMIDE COMPOUNDS Anaxis Pharma Pty Ltd (AU) 2023-06-29 WO disclosed