SCHEMBL2581014

SCHEMBL2581014

Cc1cc([N+](=O)[O-])c([N+](=O)[O-])c(C)c1C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.57
TSHR P16473 5/20 0.48
SMN1; SMN2 Q16637 1/20 0.45
ALDH1A1 P00352 5/20 0.45
TDP1 Q9NUW8 4/20 0.45
HSD17B10 Q99714 1/20 0.43
GRIN2D O15399 1/20 0.43
GRIN3B O60391 1/20 0.43
GRIN1 Q05586 1/20 0.43
GRIN2A Q12879 1/20 0.43
GRIN2B Q13224 1/20 0.43
GRIN2C Q14957 1/20 0.43
GRIN3A Q8TCU5 1/20 0.43
CYP3A4 P08684 2/20 0.42
RECQL P46063 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
GPR35 Q9HC97 2/20 0.42
MAPT P10636 2/20 0.42
HSP90AA1 P07900 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL304097 0.87 CYP1A2 (0.57) CYP1A2TSHRSMN1; SMN2ALDH1A1TDP1
SCHEMBL7527476 0.87 CYP1A2 (0.52) CYP1A2TSHRSMN1; SMN2ALDH1A1TDP1
SCHEMBL2581016 0.83 CYP1A2 (0.62) CYP1A2TSHRSMN1; SMN2ALDH1A1TDP1
SCHEMBL14020980 0.82 ALDH1A1 (0.48) CYP1A2TSHRSMN1; SMN2ALDH1A1TDP1
SCHEMBL11133854 0.82 CYP1A2 (0.67) CYP1A2TSHRSMN1; SMN2ALDH1A1TDP1
SCHEMBL20975092 0.82 CYP1A2 (0.72) CYP1A2TSHRSMN1; SMN2ALDH1A1TDP1
SCHEMBL27445177 0.82 TSHR (0.47) CYP1A2TSHRSMN1; SMN2ALDH1A1TDP1
SCHEMBL1370821 0.82 GPR35 (0.52) CYP1A2TSHRSMN1; SMN2ALDH1A1TDP1
SCHEMBL8415105 0.80 TSHR (0.50) CYP1A2TSHRSMN1; SMN2ALDH1A1TDP1
SCHEMBL9121102 0.78 CYP1A2 (0.57) CYP1A2TSHRSMN1; SMN2ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8545683-B2 Systems and methods for integrated detection Arizona Board Of Regent For And On Behalf of Arizona State University (US) 2013-10-01 US claimed
US-20110266161-A1 SYSTEMS AND METHODS FOR INTEGRATED DETECTION ARIZONA BOARD OF REGENTS FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2011-11-03 US claimed
WO-2010030874-A1 SYSTEMS AND METHODS FOR INTEGRATED DETECTION ARIZONA BOARD OF REGENTS FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2010-03-18 WO claimed
US-8545683-B2 Systems and methods for integrated detection Arizona Board Of Regent For And On Behalf of Arizona State University (US) 2013-10-01 US disclosed
US-20110266161-A1 SYSTEMS AND METHODS FOR INTEGRATED DETECTION ARIZONA BOARD OF REGENTS FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2011-11-03 US disclosed
WO-2010030874-A1 SYSTEMS AND METHODS FOR INTEGRATED DETECTION ARIZONA BOARD OF REGENTS FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2010-03-18 WO disclosed