SCHEMBL25813014

SCHEMBL25813014

CCCSc1ccc(NC)nc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 2/20 0.40
NNMT P40261 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA13 Q8N1Q1 1/20 0.39
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
AR P10275 2/20 0.33
HSD11B1 P28845 1/20 0.33
HPGD P15428 3/20 0.33
LMNA P02545 2/20 0.33
MAPK1 P28482 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
KCNH2 Q12809 2/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20196574 0.85 HCAR3 (0.42) HCAR3NNMTMAOANPC1RAB9A
SCHEMBL4248528 0.75 HCAR3 (0.46) HCAR3NNMTNPC1RAB9ALMNA
SCHEMBL25813010 0.71 CA12 (0.42) CA12CA1CA2CA7CA13
SCHEMBL13397872 0.71 CA12 (0.61) CA12CA1CA2CA7CA13
SCHEMBL17168927 0.70 AR (0.45) CA12CA1CA2CA7CA13
SCHEMBL20381749 0.70 CA12 (0.45) CA12CA1CA2CA7CA13
SCHEMBL14283230 0.69 NPC1 (0.47) HCAR3NNMTCA12CA1CA2
SCHEMBL9954024 0.69 SMN1; SMN2 (0.41) HCAR3NNMTNPC1RAB9AMAPK1
SCHEMBL11377328 0.69 MAPK1 (0.53) CA12CA1CA2CA7CA13
SCHEMBL11265059 0.69 KDM4E (0.51) CA12CA1CA2CA7CA13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3418280-B1 COMPOUNDS AS MODULATORS OF ROR GAMMA BOEHRINGER INGELHEIM INT (DE) 2023-07-12 EP disclosed