SCHEMBL25818350

SCHEMBL25818350

Nc1cnc2ccsc2c1NCC1CCN(OC(=O)c2ccccc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 9/20 0.40
ADORA2A P29274 2/20 0.35
ADORA2B P29275 2/20 0.35
CARM1 Q86X55 1/20 0.34
PRMT6 Q96LA8 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
ALDH1A1 P00352 2/20 0.33
CKS1B P61024 1/20 0.33
SKP1 P63208 1/20 0.33
SKP2 Q13309 1/20 0.33
PDGFRB P09619 1/20 0.33
KDR P35968 1/20 0.33
VNN1 O95497 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29030594 0.83 GRIN2B (0.44) GRIN2BADORA2AADORA2BCYP3A4CYP2D6
SCHEMBL25818351 0.83 NPC1 (0.35) GRIN2BADORA2AADORA2BCARM1PRMT6
SCHEMBL25256028 0.80 GRIN2B (0.65) GRIN2BCYP3A4CYP2D6CYP2C9
SCHEMBL31025943 0.80 GRIN2B (0.65) GRIN2BCYP3A4CYP2D6CYP2C9
SCHEMBL25255284 0.78 KDM4E (0.48) GRIN2BADORA2AADORA2BKDM4E
SCHEMBL31270846 0.78 KDM4E (0.48) GRIN2BADORA2AADORA2BKDM4E
SCHEMBL25818890 0.74 KCNH3 (0.41) ADORA2AADORA2BVNN1
SCHEMBL31270725 0.74 KCNH3 (0.41) ADORA2AADORA2BVNN1
SCHEMBL25424339 0.73 ALDH1A1 (0.38) ADORA2AADORA2BALDH1A1
SCHEMBL25818353 0.71 PDE4A (0.42) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125121-A1 TRICYCLIC COMPOUND, METHOD FOR PREPARING SAME, AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2023-07-06 WO disclosed