SCHEMBL25818388

SCHEMBL25818388

CCCCCc1cncc(C)n1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.47
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NOS2 P35228 1/20 0.38
HRH3 Q9Y5N1 3/20 0.33
HRH4 Q9H3N8 2/20 0.33
CYP2D6 P10635 1/20 0.33
HRH1 P35367 1/20 0.33
PPARA Q07869 1/20 0.33
TBXAS1 P24557 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL511339 0.94 NOS2 (0.43) KCNH2TDP1L3MBTL1NOS2HRH3
SCHEMBL295055 0.85 NOS1 (0.39) NOS2CYP2D6HRH1
SCHEMBL10834770 0.83 CYP2D6 (0.38) NOS2CYP2D6HRH1
SCHEMBL4685578 0.81 KCNH2 (0.32) KCNH2CYP2D6HRH1
SCHEMBL22877896 0.79 CYP2D6 (0.34) TDP1CYP2D6HRH1MEN1KMT2A
SCHEMBL22616936 0.78 KCNH2 (0.46) KCNH2TDP1L3MBTL1NOS2HRH3
SCHEMBL23138935 0.78 KCNH2 (0.35) KCNH2
SCHEMBL105987 0.76
SCHEMBL5302424 0.75 CYP2D6 (0.35) NOS2CYP2D6HRH1MEN1KMT2A
SCHEMBL24618582 0.75 HRH4 (0.36) TDP1NOS2HRH3HRH4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131868-A1 HETEROCYCLIC INHIBITORS OF GLUT9 FOR TREATMENT OF DISEASE HORIZON THERAPEUTICS IRELAND DAC (IE) 2023-07-13 WO disclosed