SCHEMBL25818907

SCHEMBL25818907

CC1CC(Nc2nc(NCc3ccc(C#N)cc3)nc3ccccc23)=NN1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 9/20 0.60
CTNNB1 P35222 1/20 0.48
TCF7L2 Q9NQB0 1/20 0.48
USP1 O94782 1/20 0.46
WDR48 Q8TAF3 1/20 0.46
RAD52 P43351 1/20 0.46
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
PKM P14618 1/20 0.45
UBE2N P61088 1/20 0.45
KMT2A Q03164 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
RCE1 Q9Y256 1/20 0.45
BCHE P06276 3/20 0.44
ACHE P22303 3/20 0.44
APP P05067 2/20 0.44
GRK6 P43250 1/20 0.43
MERTK Q12866 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25818900 0.87 NTRK1 (0.58) NTRK1RAD52KDM4EALDH1A1LMNA
SCHEMBL25818886 0.87 NTRK1 (0.58) NTRK1CTNNB1TCF7L2RAD52KDM4E
SCHEMBL2203869 0.76 NTRK1 (0.67) NTRK1CTNNB1TCF7L2USP1WDR48
SCHEMBL25818909 0.75 NTRK1 (1.00) NTRK1GRK6PLK4
SCHEMBL31471730 0.74 NTRK1 (0.79) NTRK1
SCHEMBL20352461 0.74 LMNA (0.40) ALDH1A1LMNAMAPTKMT2A
SCHEMBL2204282 0.73 NTRK1 (0.63) NTRK1CTNNB1TCF7L2USP1WDR48
SCHEMBL22054938 0.73 WHR1 (0.46) LMNAMAPTKMT2ANPSR1BCHE
SCHEMBL21567312 0.72 ACHE (0.77) NTRK1CTNNB1TCF7L2USP1WDR48
SCHEMBL30092903 0.72 ACHE (0.77) NTRK1CTNNB1TCF7L2USP1WDR48

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023123883-A1 METHOD FOR PREPARING QUINAZOLINE DERIVATIVE AND ANALOG THEREOF AND USE THEREOF 沈阳药科大学 2023-07-06 WO disclosed