SCHEMBL2582189

SCHEMBL2582189

COC(=O)c1ccc2c(c1)CC(C)(C)C(c1cccc(C(=O)N(C)C3CNC3)c1)N2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.40
CHRNA4 P43681 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.38
ALDH1A1 P00352 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 3/20 0.34
MAPT P10636 3/20 0.34
GAA P10253 1/20 0.34
MAPK1 P28482 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
RAB9A P51151 2/20 0.34
NPC1 O15118 1/20 0.34
TSHR P16473 1/20 0.34
F10 P00742 1/20 0.33
F11 P03951 1/20 0.33
F7 P08709 1/20 0.33
SLC10A2 Q12908 1/20 0.33
AR P10275 1/20 0.33
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2534306 0.86 CHRNB2 (0.38) CHRNB2CHRNA4SMN1; SMN2ALDH1A1MEN1
SCHEMBL2533556 0.83 ALDH1A1 (0.41) CHRNB2CHRNA4SMN1; SMN2ALDH1A1MEN1
SCHEMBL2532907 0.83 AR (0.44) SMN1; SMN2ALDH1A1MEN1KMT2AKDM4E
SCHEMBL2530168 0.83 ALDH1A1 (0.43) CHRNB2CHRNA4SMN1; SMN2ALDH1A1MEN1
SCHEMBL2533076 0.83 MEN1 (0.37) CHRNB2CHRNA4SMN1; SMN2ALDH1A1MEN1
SCHEMBL2533058 0.82 MEN1 (0.40) CHRNB2CHRNA4SMN1; SMN2ALDH1A1MEN1
SCHEMBL2531587 0.81 ABL1 (0.40) SMN1; SMN2ALDH1A1MEN1KMT2AMAPT
SCHEMBL2535580 0.81 ROCK2 (0.36) SMN1; SMN2ALDH1A1MEN1KMT2ATSHR
SCHEMBL2535027 0.81 ALDH1A1 (0.44) SMN1; SMN2ALDH1A1MEN1KMT2AKDM4E
SCHEMBL2533669 0.81 ALDH1A1 (0.41) CHRNB2CHRNA4SMN1; SMN2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2558449-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2013-02-20 EP disclosed
WO-2011128251-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-10-20 WO disclosed