SCHEMBL25826817

SCHEMBL25826817

Cn1cc(Br)c(COCCNC(=O)OC(C)(C)C)n1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.41
ADORA1 P30542 6/20 0.41
ADORA3 P0DMS8 5/20 0.41
CA12 O43570 5/20 0.40
CA1 P00915 5/20 0.40
CA2 P00918 5/20 0.40
CA9 Q16790 5/20 0.40
ALDH1A1 P00352 1/20 0.38
GFER P55789 1/20 0.38
IDO1 P14902 1/20 0.37
SUV39H2 Q9H5I1 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
ADORA2B P29275 1/20 0.35
DRD2 P14416 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24553575 0.85 ALDH1A1 (0.46) ADORA2AADORA1ADORA3CA12CA1
SCHEMBL29456690 0.82 KDM4E (0.44) CA12CA1CA2CA9ALDH1A1
SCHEMBL25826819 0.79 PPARA (0.37) CA1CA2CA9ALDH1A1
SCHEMBL25424201 0.79 TP53 (0.33) ALDH1A1
SCHEMBL31465653 0.78 SSTR4 (0.34)
SCHEMBL24192223 0.77 CA12 (0.48) ADORA2AADORA1ADORA3CA12CA1
SCHEMBL24192594 0.76 CA12 (0.40) CA12CA1CA2CA9ALDH1A1
SCHEMBL25471683 0.73 CTSS (0.48) CA12CA1CA2CA9IDO1
SCHEMBL25056245 0.73 ALDH1A1 (0.46) ADORA2AADORA1ADORA3ALDH1A1GFER
SCHEMBL25301986 0.72 IDO1 (0.47) CA12CA1CA2CA9IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023133375-A1 MACROCYCLIC COMPOUNDS AND USE AS KINASE INHIBITORS BLOSSOMHILL THERAPEUTICS, INC. (US) 2023-07-13 WO disclosed