SCHEMBL25828656

SCHEMBL25828656

CCCCCc1ccc(S(=O)(=O)Nc2cc(-c3csc(N)n3)ccc2N2CCN(C)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NMT1 P30419 1/20 0.44
HTR2A P28223 3/20 0.44
HTR2C P28335 3/20 0.44
HTR2B P41595 1/20 0.44
DRD2 P14416 3/20 0.43
DRD3 P35462 3/20 0.43
HTR6 P50406 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
AKT1 P31749 6/20 0.41
ALDH1A1 P00352 2/20 0.41
PDPK1 O15530 1/20 0.41
ABCB11 O95342 1/20 0.41
AKT2 P31751 1/20 0.41
GAB1 Q13480 1/20 0.41
AKT3 Q9Y243 1/20 0.41
NPC1 O15118 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18425498 0.87 ALDH1A1 (0.48) NMT1CYP3A4AKT1ALDH1A1PDPK1
SCHEMBL22590668 0.87 PHGDH (0.46) NMT1HTR2AHTR2CDRD2DRD3
SCHEMBL25735584 0.85 SMN1; SMN2 (0.45) NMT1CYP3A4ALDH1A1NPC1RAB9A
SCHEMBL25250241 0.85 SMN1; SMN2 (0.47) NMT1CYP3A4ALDH1A1NPC1RAB9A
SCHEMBL25828673 0.82 SMN1; SMN2 (0.44) NMT1CYP3A4ALDH1A1NPC1RAB9A
SCHEMBL25237942 0.81 SMN1; SMN2 (0.48) AKT1ALDH1A1PDPK1ABCB11AKT2
SCHEMBL30479932 0.81 SMN1; SMN2 (0.48) AKT1ALDH1A1PDPK1ABCB11AKT2
SCHEMBL25735583 0.80 ALDH1A1 (0.45) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL18424453 0.79 ALDH1A1 (0.50) CYP3A4ALDH1A1NPC1RAB9AMEN1
SCHEMBL22590669 0.79 ALDH1A1 (0.46) CYP3A4AKT1ALDH1A1PDPK1ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4201928-A1 BENZENE SULFONAMIDE THIAZOLE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF CANCERS Institut National de la Santé et de la Recherche Médicale (INSERM) (FR) 2023-06-28 EP disclosed