SCHEMBL258365

SCHEMBL258365

COc1ccc(N)c(C(N)=O)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 2/20 0.57
PARP1 P09874 2/20 0.52
PARP10 Q53GL7 2/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
PARP2 Q9UGN5 1/20 0.52
PARP4 Q9UKK3 1/20 0.52
KDM4E B2RXH2 3/20 0.51
ALDH1A1 P00352 3/20 0.50
CYP3A4 P08684 2/20 0.50
IKBKB O14920 2/20 0.49
MAPT P10636 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
MEN1 O00255 1/20 0.48
GAA P10253 1/20 0.48
THRB P10828 1/20 0.48
RECQL P46063 1/20 0.48
BLM P54132 1/20 0.48
KMT2A Q03164 1/20 0.48
MCL1 Q07820 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30821626 1.00 NOS2 (0.57) NOS2PARP1PARP10CA1CA2
Hydrochloric Acid SCHEMBL11466167 0.98 NOS2 (0.56) NOS2PARP1PARP10CA1CA2
SCHEMBL5306467 0.86 IKBKB (0.65) NOS2PARP1PARP10CA1CA2
SCHEMBL221141 0.85 SMN1; SMN2 (0.59) NOS2KDM4EALDH1A1CYP3A4MAPT
SCHEMBL632502 0.85 ALDH1A1 (0.59) NOS2KDM4EALDH1A1CYP3A4MAPT
SCHEMBL29923727 0.85 ALDH1A1 (0.59) NOS2KDM4EALDH1A1CYP3A4MAPT
SCHEMBL29380973 0.85 SMN1; SMN2 (0.59) NOS2KDM4EALDH1A1CYP3A4MAPT
SCHEMBL148855 0.85 ALDH1A1 (0.53) NOS2PARP1PARP10CA1CA2
SCHEMBL27720018 0.85 SMN1; SMN2 (0.59) NOS2KDM4EALDH1A1CYP3A4MAPT
SCHEMBL25328315 0.84 NR4A1 (0.52) NOS2PARP10PARP2PARP4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 217 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122010957-A Preparation method of fullerene pyrrolidine quinazolinone 湖北大学 2026-05-12 CN claimed
CN-117820337-A Preparation method of 12H-benzo [4,5] thiazolo [2,3-b ] quinazoline 12-ketone compound 赣南师范大学 2024-04-05 CN claimed
CN-111848527-A 4-chloro-2- (2-fluoro-4-methoxyphenyl) -6-methoxyquinazoline and synthetic method thereof 南通大学 2020-10-30 CN claimed
CN-122010957-A Preparation method of fullerene pyrrolidine quinazolinone 湖北大学 2026-05-12 CN disclosed
EP-4731216-A1 HETEROARYL-AMINE COMPOUNDS AND USE THEREOF AS HDAC6 INHIBITORS Augustine Therapeutics (BE) 2026-04-29 EP disclosed
EP-4719394-A2 INHIBITORS OF TYK2 Atomwise Inc. (US) 2026-04-08 EP disclosed
US-20260048051-A1 TREATMENT OF INFLAMMATORY BOWEL DISEASE ATOMWISE INC (US) 2026-02-19 US disclosed
EP-4127157-B1 MODIFIED DIPEPTIDE CLEAVASES, USES THEREOF AND RELATED KITS ENCODIA INC (US) 2026-02-11 EP disclosed
WO-2025227032-A1 METHODS FOR DEGRADATION OF CYCLIN K AND INHIBITION OF CYCLIN DEPENDENT KINASES REMIX THERAPEUTICS INC. (US) 2025-10-30 WO disclosed
US-12421222-B2 Substituted quinazolines as HDAC6 inhibitors AUGUSTINE THERAPEUTICS (BE) 2025-09-23 US disclosed
US-12358904-B2 Inhibitors of TYK2 Atomwise Inc. (US) 2025-07-15 US disclosed
US-6608056-B1 Phosphatidylinositol 3-kinase inhibitors and carcinostatic agents YAMANOUCHI PHARMACEUTICAL CO., LTD (JP) 2003-08-19 US disclosed
CN-1426398-A Fused heteroaryl derivatives YAMANOUCHI PHARMA CO LTD (JP) 2003-06-25 CN disclosed
EP-1277738-A1 CONDENSED HETEROARYL DERIVATIVES YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 2003-01-22 EP disclosed
US-6479499-B1 INHIBITORS OF TUBULIN POLYMERIZATION NATIONAL SCIENCE COUNCIL (TW) 2002-11-12 US disclosed
US-20020151544-A1 Fused heteroaryl derivatives ASTELLAS PHARMA INC. (JP) 2002-10-17 US disclosed
US-5030727-A Reacting an anthronilide derivative with a thiazole derivative or a fluorozuinazolone with a neucleophile BASF AKTIENGESELLSCHAFT (DE) 1991-07-09 US disclosed
EP-0263523-A2 Process for the preparation of thiazolo [2,3-b] quinazolones BASF Aktiengesellschaft (DE) 1988-04-13 EP disclosed
US-4400507-A FOR COLORING POLYMERS, LACQUERS CIBA-GEIGY CORPORATION (US) 1983-08-23 US disclosed
US-4262120-A YELLOW TO ORANGE SHADES OF GOOD FASTNESS CIBA-GEIGY CORPORATION (US) 1981-04-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260048051-A1 TREATMENT OF INFLAMMATORY BOWEL DISEASE TYK2, FRK, DYRK2 NOS2 1750/4885PARP1 2186/4885PARP10 2377/4885
US-12358904-B2 Inhibitors of TYK2 TYK2, LCK, JAK2 NOS2 3388/4885PARP1 1129/4885PARP10 501/4885
US-20020151544-A1 Fused heteroaryl derivatives PIK3CD, PIK3R3, PIK3C2A NOS2 3761/4885PARP1 1165/4885PARP10 1139/4885
US-12421222-B2 Substituted quinazolines as HDAC6 inhibitors HDAC6, HDAC9, HDAC1 NOS2 3273/4885PARP1 541/4885PARP10 624/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.