SCHEMBL148855

SCHEMBL148855

COc1ccc(C(N)=O)c(N)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.53
KDM4E B2RXH2 3/20 0.53
MEN1 O00255 2/20 0.53
MAPT P10636 2/20 0.53
THRB P10828 2/20 0.53
KMT2A Q03164 2/20 0.53
GAA P10253 2/20 0.53
RECQL P46063 1/20 0.53
BLM P54132 1/20 0.53
MCL1 Q07820 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
PARP1 P09874 2/20 0.52
PARP10 Q53GL7 2/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
PARP2 Q9UGN5 1/20 0.52
PARP4 Q9UKK3 1/20 0.52
NPC1 O15118 2/20 0.52
RAB9A P51151 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nitrogen SCHEMBL8706863 0.96 PARP1 (0.51) ALDH1A1KDM4EMEN1MAPTTHRB
SCHEMBL9929149 0.86 NPC1 (0.63) ALDH1A1KDM4EMEN1MAPTTHRB
SCHEMBL147211 0.85 SMN1; SMN2 (0.54) ALDH1A1KDM4EMEN1MAPTTHRB
SCHEMBL312677 0.85 ALDH1A1 (0.65) ALDH1A1KDM4EMEN1MAPTTHRB
SCHEMBL29976235 0.85 ALDH1A1 (0.65) ALDH1A1KDM4EMEN1MAPTTHRB
SCHEMBL258365 0.85 NOS2 (0.57) ALDH1A1KDM4EMEN1MAPTTHRB
SCHEMBL30821626 0.85 NOS2 (0.57) ALDH1A1KDM4EMEN1MAPTTHRB
SCHEMBL2835948 0.84 PARP1 (0.55) ALDH1A1KDM4EMAPTGAASMN1; SMN2
Hydrochloric Acid SCHEMBL11466167 0.83 NOS2 (0.56) ALDH1A1KDM4EMEN1MAPTTHRB
Hydrochloric Acid SCHEMBL30735974 0.83 ALDH1A1 (0.62) ALDH1A1KDM4EMEN1MAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 171 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9068989-B2 Reagent system and method LEICA BIOSYSTEMS MELBOURNE PTY LTD (AU) 2015-06-30 US claimed
US-20120208287-A1 REAGENT SYSTEM AND METHOD LEICA BIOSYSTEMS MELBOURNE PTY LTD. (AU) 2012-08-16 US claimed
EP-2459983-A1 REAGENT SYSTEM AND METHOD Leica Biosystems Melbourne Pty Ltd (AU) 2012-06-06 EP claimed
WO-2011011826-A1 REAGENT SYSTEM AND METHOD LEICA BIOSYSTEMS MELBOURNE PTY LTD (AU) 2011-02-03 WO claimed
US-20060035939-A1 3-Aminobenzamide compounds and inhibitors of vanilloid receptor subtype 1 (VR1) activity JAPAN TOBACCO INC. (JP) 2006-02-16 US claimed
EP-4127157-B1 MODIFIED DIPEPTIDE CLEAVASES, USES THEREOF AND RELATED KITS ENCODIA INC (US) 2026-02-11 EP disclosed
US-20250171447-A1 ADENOSINE RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS AND THEIR USE THEREOF MERCK SHARP & DOHME LLC (US) 2025-05-29 US disclosed
EP-4479056-A1 ADENOSINE RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS AND THEIR USE THEREOF Merck Sharp & Dohme LLC (US) 2024-12-25 EP disclosed
EP-2408454-B1 NOVEL ANTI-INFLAMMATORY AGENTS RESVERLOGIX CORP (CA) 2024-07-24 EP disclosed
US-20240011009-A1 MODIFIED DIPEPTIDE CLEAVASES, USES THEREOF AND RELATED KITS Encodia, Inc. (US) 2024-01-11 US disclosed
US-11788080-B2 Modified cleavases, uses thereof and related kits Encodia, Inc. (US) 2023-10-17 US disclosed
WO-2023158626-A1 ADENOSINE RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS AND THEIR USE THEREOF MERCK SHARP & DOHME LLC (US) 2023-08-24 WO disclosed
US-4160100-A OXAMIC ACID DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 1979-07-03 US disclosed
US-4154961-A Oxamic acid derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1979-05-15 US disclosed
US-4069343-A OXAMIC ACID DERIVATIVES FOR THE PREVENTION OF IMMEDIATE TYPE HYPERSENSITIVITY REACTIONS AMERICAN HOME PRODUCTS CORPORATION (US) 1978-01-17 US disclosed
US-4054661-A Pyridyl oxamic acid derivatives and use in the prevention of allergic reactions AMERICAN HOME PRODUCTS CORPORATION (US) 1977-10-18 US disclosed
US-4054666-A Compositions and methods of treating immediate hypersensitivity reactions with thiazolyl oxamic acid derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1977-10-18 US disclosed
US-4054657-A Pyrimidinyl oxamic acids and esters, and compositions and methods for the suppression of allergic manifestations AMERICAN HOME PRODUCTS CORPORATION (US) 1977-10-18 US disclosed
US-4036837-A 2 Alkoxyoxamoyl-pyrazines AMERICAN HOME PRODUCTS CORPORATION (US) 1977-07-19 US disclosed
US-3966965-A Oxamic acid derivatives for the prevention of immediate type hypersensitivity reactions AMERICAN HOME PRODUCTS CORPORATION (US) 1976-06-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250171447-A1 ADENOSINE RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS AND THEIR USE THEREOF ADORA2A, ADORA2B, ADORA1 ALDH1A1 483/4885KDM4E 3489/4885MEN1 2390/4885
US-20060035939-A1 3-Aminobenzamide compounds and inhibitors of vanilloid receptor subtype 1 (VR1) activity TRPV1, TRPV6, TRPV3 ALDH1A1 1481/4885KDM4E 3049/4885MEN1 3079/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.