SCHEMBL2583768

SCHEMBL2583768

COc1ccccc1Nc1nc(NCc2ccccc2)c2ccccc2n1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 3/20 0.71
HTT P42858 2/20 0.71
TSHR P16473 2/20 0.71
USP2 O75604 1/20 0.71
MAPK1 P28482 3/20 0.71
KDM4E B2RXH2 3/20 0.71
MAPT P10636 3/20 0.71
NPSR1 Q6W5P4 3/20 0.71
RECQL P46063 1/20 0.71
SLC2A1 P11166 2/20 0.69
KMT2A Q03164 2/20 0.67
MEN1 O00255 1/20 0.67
GAA P10253 1/20 0.67
BLM P54132 1/20 0.67
LMNA P02545 2/20 0.63
CYP1A2 P05177 1/20 0.63
CYP3A4 P08684 1/20 0.63
CYP2D6 P10635 1/20 0.63
CYP2C19 P33261 1/20 0.63
SMN1; SMN2 Q16637 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2593560 0.89 SLC2A1 (0.60) RAD52HTTTSHRUSP2MAPK1
SCHEMBL12176124 0.87 KMT2A (0.65) RAD52HTTTSHRUSP2MAPK1
SCHEMBL10031967 0.84 RAD52 (0.98) RAD52HTTTSHRUSP2MAPK1
SCHEMBL12175940 0.84 SLC2A1 (0.70) RAD52TSHRUSP2MAPK1KDM4E
SCHEMBL14281045 0.84 SLC2A1 (0.73) RAD52HTTMAPK1KDM4EMAPT
SCHEMBL12175851 0.83 SLC2A1 (0.61) RAD52HTTTSHRMAPK1KDM4E
SCHEMBL2583400 0.83 SLC2A1 (0.61) RAD52HTTTSHRMAPK1KDM4E
SCHEMBL30933352 0.82 RAD52 (1.00) RAD52HTTTSHRUSP2MAPK1
SCHEMBL18282619 0.82 RAD52 (1.00) RAD52HTTTSHRUSP2MAPK1
SCHEMBL8900319 0.82 NPY5R (0.67) RAD52HTTTSHRUSP2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2566480-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE California Institute of Technology (US) 2013-03-13 EP disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed