SCHEMBL2583769

SCHEMBL2583769

CSc1ccc(CCCCCNc2ccc3[nH]cnc3c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QPCT Q16769 8/20 0.43
QPCTL Q9NXS2 1/20 0.43
RAB9A P51151 4/20 0.37
NPC1 O15118 3/20 0.37
MAPT P10636 3/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
EPHX1 P07099 1/20 0.36
POLA1 P09884 2/20 0.35
PIK3CD O00329 1/20 0.35
CDC7 O00311 1/20 0.35
DBF4 Q9UBU7 1/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
HPGD P15428 1/20 0.34
RECQL P46063 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2545579 0.83 RAB9A (0.55) QPCTQPCTLRAB9ANPC1MAPT
SCHEMBL2547500 0.76 EPHX1 (0.47) CYP1A2CYP2C19CYP3A4CYP2D6EPHX1
SCHEMBL2541353 0.74 QPCT (0.54) QPCTQPCTLPIK3CD
SCHEMBL20011724 0.73 EPHX1 (0.43) QPCTMAPTEPHX1RECQL
SCHEMBL1976000 0.71 QPCT (0.45) QPCTQPCTLMAPTHPGDRECQL
SCHEMBL2539456 0.71 QPCT (0.74) QPCTQPCTLMAPTCDC7DBF4
SCHEMBL18126690 0.70 MMP12 (0.41) QPCTMAPTEPHX1RECQL
SCHEMBL8733538 0.70 QPCT (0.44) QPCTQPCTLMAPTHPGDRECQL
SCHEMBL9224383 0.69 HTR1A (0.48) QPCTRAB9AMAPTCYP3A4EPHX1
SCHEMBL2538614 0.69 NPC1 (0.56) QPCTRAB9ANPC1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2560953-A2 NOVEL INHIBITORS Probiodrug AG (DE) 2013-02-27 EP disclosed
WO-2011131748-A2 NOVEL INHIBITORS PROBIODRUG AG (DE) 2011-10-27 WO disclosed