SCHEMBL2583780

SCHEMBL2583780

Fc1cccc(Nc2nc(NCc3ccccc3)c3ccccc3n2)c1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.67
RAD52 P43351 1/20 0.64
KMT2A Q03164 4/20 0.63
KDM4E B2RXH2 3/20 0.63
MAPT P10636 2/20 0.63
NPSR1 Q6W5P4 2/20 0.63
ALDH1A1 P00352 1/20 0.63
LMNA P02545 1/20 0.63
PKM P14618 1/20 0.63
UBE2N P61088 1/20 0.63
RCE1 Q9Y256 1/20 0.63
APP P05067 3/20 0.61
SLC2A1 P11166 1/20 0.61
MEN1 O00255 2/20 0.60
NPC1 O15118 1/20 0.60
TP53 P04637 1/20 0.60
ALOX15 P16050 1/20 0.60
TSHR P16473 1/20 0.60
RAB9A P51151 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2584997 0.89 SOS1 (0.65) PDE5ARAD52KMT2AKDM4EMAPT
SCHEMBL2580376 0.87 RAD52 (0.76) RAD52KMT2AKDM4EMAPTNPSR1
SCHEMBL3640101 0.87 RAD52 (0.79) PDE5ARAD52KMT2AKDM4EMAPT
SCHEMBL2588903 0.85 SOS1 (0.72) PDE5ARAD52KMT2AKDM4EMAPT
SCHEMBL12176293 0.85 SOS1 (0.72) PDE5ARAD52KMT2AKDM4EMAPT
SCHEMBL2590904 0.85 PDE5A (0.67) PDE5ARAD52KMT2AKDM4EMAPT
SCHEMBL2583209 0.85 SOS1 (0.72) PDE5ARAD52KMT2AKDM4EMAPT
SCHEMBL2590218 0.85 SOS1 (0.66) PDE5ARAD52KMT2AKDM4EMAPT
SCHEMBL2583406 0.85 PDE5A (0.64) PDE5ARAD52KMT2AKDM4EMAPT
SCHEMBL2590870 0.85 SLC2A1 (0.60) PDE5ARAD52KMT2AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2566480-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE California Institute of Technology (US) 2013-03-13 EP disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed