SCHEMBL12176293

SCHEMBL12176293

Cc1cccc(Nc2nc(NCc3ccccc3)c3ccccc3n2)c1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 1/20 0.72
MAPT P10636 3/20 0.71
NPSR1 Q6W5P4 3/20 0.71
ALDH1A1 P00352 2/20 0.71
LMNA P02545 2/20 0.71
KMT2A Q03164 2/20 0.71
USP2 O75604 1/20 0.71
HPGD P15428 1/20 0.71
NR2F2 P24468 1/20 0.71
MAPK1 P28482 1/20 0.71
SMN1; SMN2 Q16637 1/20 0.71
PDE5A O76074 2/20 0.67
RAD52 P43351 1/20 0.64
SLC2A1 P11166 2/20 0.64
KDM4E B2RXH2 1/20 0.63
PKM P14618 1/20 0.63
UBE2N P61088 1/20 0.63
RCE1 Q9Y256 1/20 0.63
BCHE P06276 4/20 0.62
ACHE P22303 4/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2587460 0.89 SOS1 (0.65) SOS1MAPTNPSR1ALDH1A1LMNA
SCHEMBL12175983 0.87 RAD52 (0.76) MAPTNPSR1ALDH1A1LMNAKMT2A
SCHEMBL3640101 0.87 RAD52 (0.79) MAPTNPSR1ALDH1A1LMNAKMT2A
SCHEMBL12175981 0.86 SLC2A1 (0.76) MAPTNPSR1ALDH1A1LMNAKMT2A
SCHEMBL2588903 0.85 SOS1 (0.72) SOS1MAPTNPSR1ALDH1A1LMNA
SCHEMBL2590904 0.85 PDE5A (0.67) MAPTNPSR1ALDH1A1LMNAKMT2A
SCHEMBL2583780 0.85 PDE5A (0.67) MAPTNPSR1ALDH1A1LMNAKMT2A
SCHEMBL2583209 0.85 SOS1 (0.72) SOS1MAPTNPSR1ALDH1A1LMNA
SCHEMBL2588902 0.85 SOS1 (0.66) SOS1MAPTNPSR1ALDH1A1LMNA
SCHEMBL2590870 0.85 SLC2A1 (0.60) SOS1MAPTNPSR1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed