SCHEMBL2590218

SCHEMBL2590218

Fc1ccc(CNc2nc(Nc3cccc(Cl)c3)nc3ccccc23)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 2/20 0.66
PDE5A O76074 4/20 0.59
MAPT P10636 3/20 0.56
KMT2A Q03164 3/20 0.56
LMNA P02545 2/20 0.56
MEN1 O00255 1/20 0.56
APP P05067 1/20 0.56
ABCG2 Q9UNQ0 1/20 0.55
CTNNB1 P35222 1/20 0.55
TCF7L2 Q9NQB0 1/20 0.55
MERTK Q12866 1/20 0.55
NTRK1 P04629 2/20 0.54
KDM4E B2RXH2 2/20 0.54
NPSR1 Q6W5P4 2/20 0.54
XBP1 P17861 1/20 0.54
MAPK1 P28482 1/20 0.54
RAD52 P43351 1/20 0.54
KCNH3 Q9ULD8 1/20 0.54
ALDH1A1 P00352 1/20 0.53
PKM P14618 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2588890 0.92 SOS1 (0.70) SOS1PDE5AMAPTKMT2ALMNA
SCHEMBL2583209 0.92 SOS1 (0.72) SOS1PDE5AMAPTKMT2ALMNA
SCHEMBL2584997 0.90 SOS1 (0.65) SOS1PDE5AMAPTKMT2ALMNA
SCHEMBL2588902 0.89 SOS1 (0.66) SOS1PDE5AMAPTKMT2ALMNA
SCHEMBL2587225 0.89 SOS1 (0.66) SOS1PDE5AMAPTKMT2ALMNA
SCHEMBL2592287 0.89 SOS1 (0.71) SOS1PDE5AMAPTKMT2ALMNA
SCHEMBL2590586 0.86 SLC2A1 (0.73) SOS1PDE5ALMNAAPPCTNNB1
SCHEMBL4738601 0.86 RAD52 (0.62) SOS1PDE5AMAPTKMT2ALMNA
SCHEMBL2583780 0.85 PDE5A (0.67) PDE5AMAPTKMT2ALMNAMEN1
SCHEMBL2590962 0.85 SOS1 (0.66) SOS1PDE5AMAPTKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2566480-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE California Institute of Technology (US) 2013-03-13 EP disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed