SCHEMBL258406

SCHEMBL258406

CCCCCCCC(=O)NCCS(=O)(=O)O

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CASP2 P42575 1/20 0.61
FAAH O00519 5/20 0.61
NAAA Q02083 1/20 0.58
DNM1 Q05193 2/20 0.57
EPHX2 P34913 4/20 0.54
SLC6A5 Q9Y345 2/20 0.53
ALDH1A1 P00352 2/20 0.51
SELP P16109 1/20 0.50
HSP90AA1 P07900 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL258718 1.00 CASP2 (0.61) CASP2FAAHNAAADNM1EPHX2
SCHEMBL11051906 1.00 CASP2 (0.61) CASP2FAAHNAAADNM1EPHX2
SCHEMBL11228741 1.00 CASP2 (0.61) CASP2FAAHNAAADNM1EPHX2
SCHEMBL258662 1.00 CASP2 (0.61) CASP2FAAHNAAADNM1EPHX2
SCHEMBL6856630 1.00 CASP2 (0.61) CASP2FAAHNAAADNM1EPHX2
SCHEMBL10882190 1.00 CASP2 (0.61) CASP2FAAHNAAADNM1EPHX2
SCHEMBL233312 1.00 CASP2 (0.61) CASP2FAAHNAAADNM1EPHX2
SCHEMBL258527 1.00 CASP2 (0.61) CASP2FAAHNAAADNM1EPHX2
SCHEMBL21274180 1.00 CASP2 (0.61) CASP2FAAHNAAADNM1EPHX2
SCHEMBL31510848 1.00 CASP2 (0.61) CASP2FAAHNAAADNM1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 267 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260043065-A1 Methods of Administering 3,4-Diaminopyridine SERB SA (BE) 2026-02-12 US disclosed
US-20240316050-A1 TREATMENT OF DISORDERS ASSOCIATED WITH LOW BH4 BIOAVAILABILITY OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2024-09-26 US disclosed
US-11873525-B2 Methods of administering 3,4-diaminopridine SERB SA (BE) 2024-01-16 US disclosed
US-11845977-B2 Methods of administering 3,4-diaminopridine SERB SA (BE) 2023-12-19 US disclosed
US-11840515-B2 Methods for preparing N-(4-fluorobenzyl)-N-(1-methylpiperidin-4-yl)-N′-(4-(2-methylpropyloxy)phenylmethyl)carbamide and its tartrate salt and polymorphic form c ACADIA PHARMACEUTICALS INC. (US) 2023-12-12 US disclosed
EP-4262806-A1 TREATMENT OF DISORDERS ASSOCIATED WITH LOW BH4 BIOAVAILABILITY Oxford University Innovation Limited (GB) 2023-10-25 EP disclosed
US-20230313265-A1 Methods of Administering 3,4-Diaminopridine SERB SA (BE) 2023-10-05 US disclosed
US-20230295685-A1 Methods of Administering 3,4-Diaminopridine SERB SA (BE) 2023-09-21 US disclosed
CN-116723842-A Treatment of conditions associated with low BH4 bioavailability 牛津大学科技创新有限公司 2023-09-08 CN disclosed
US-20230034700-A1 Methods of Administering 3,4-Diaminopyridine SERB SA (BE) 2023-02-02 US disclosed
EP-1595880-A1 Crystalline forms of a pyridinyl-sulfonamide and their use as endothelin receptor antagonists Speedel Pharma AG (CH) 2005-11-16 EP disclosed
WO-2005065018-A2 CRYSTALLINE FORMS OF (6R) -L-ERYTHRO-TETRAHYDROBIOPTERIN DIHYDROCHLORIDE MERCK EPROVA AG (US) 2005-07-21 WO disclosed
US-20050147629-A1 Pharmaceutical formulation comprising non-peptide renin inhibitor and surfactant NODEN PHARMA DAC (IE) 2005-07-07 US disclosed
WO-2005058872-A1 CRYSTALLINE FORMS OF (+)- AND (-)-ERYTHRO-MEFLOQUINE HYDROCHLORIDE ARAKIS LTD. (GB) 2005-06-30 WO disclosed
WO-2005049000-A2 TREATMENT OF PHENYLKETONURIAS WITH BH4 BIOMARIN PHARMACEUTICAL INC. (US) 2005-06-02 WO disclosed
EP-1517682-A1 PHARMACEUTICAL FORMULATION COMPRISING NON-PEPTIDE RENIN INHIBITOR AND SURFACTANT Speedel Pharma AG (CH) 2005-03-30 EP disclosed
US-20040077232-A1 Pharmaceutical compositions EBNER ANDREAS (DE) 2004-04-22 US disclosed
WO-2004002466-A1 PHARMACEUTICAL FORMULATION COMPRISING NON-PEPTIDE RENIN INHIBITOR AND SURFACTANT SPEEDEL PHARMA AG (CH) 2004-01-08 WO disclosed
EP-1372611-A2 PHARMACEUTICAL COMPOSITION COMPRISING A POORLY WATER-SOLUBLE ACTIVE INGREDIENT, A SURFACTANT AND A WATER-SOLUBLE POLYMER Novartis AG (CH) 2004-01-02 EP disclosed
WO-2002076432-A2 PHARMACEUTICAL COMPOSITION COMPRISING A POORLY WATER-SOLUBLE ACTIVE INGREDIENT, A SURFACTANT AND A WATER-SOLUBLE POLYMER NOVARTIS AG (CH) 2002-10-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230295685-A1 Methods of Administering 3,4-Diaminopridine NAT1, SAT1, AADAC CASP2 3524/4885FAAH 1128/4885NAAA 83/4885
US-11840515-B2 Methods for preparing N-(4-fluorobenzyl)-N-(1-methylpiperidin-4-yl)-N′-(4-(2-methylpropyloxy)phenylmethyl)carbamide and its tartrate salt and polymorphic form c NR3C2, NR2C2, CYP4A22 CASP2 4386/4885FAAH 4301/4885NAAA 3156/4885
US-20260043065-A1 Methods of Administering 3,4-Diaminopyridine NAT1, SAT1, NANS CASP2 3117/4885FAAH 2280/4885NAAA 318/4885
US-20230313265-A1 Methods of Administering 3,4-Diaminopridine NAT1, SAT1, AADAC CASP2 3524/4885FAAH 1128/4885NAAA 83/4885
US-11873525-B2 Methods of administering 3,4-diaminopridine NAT1, SAT1, AADAC CASP2 3524/4885FAAH 1128/4885NAAA 83/4885
US-11845977-B2 Methods of administering 3,4-diaminopridine NAT1, SAT1, AADAC CASP2 3524/4885FAAH 1128/4885NAAA 83/4885
US-20230034700-A1 Methods of Administering 3,4-Diaminopyridine NAT1, NAT10, SAT1 CASP2 3368/4885FAAH 1374/4885NAAA 66/4885
US-20050147629-A1 Pharmaceutical formulation comprising non-peptide renin inhibitor and surfactant REN, AGT, ACE CASP2 3177/4885FAAH 529/4885NAAA 983/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.