SCHEMBL25840688

SCHEMBL25840688

O=C(Cc1cccnc1)Nc1nc(CC(O)N2CCC(N3CCCC3)CC2)cs1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.47
NAMPT P43490 2/20 0.41
HTT P42858 1/20 0.40
CTPS1 P17812 1/20 0.40
MAPT P10636 1/20 0.40
GLS O94925 3/20 0.39
SIGMAR1 Q99720 1/20 0.39
ROCK1 Q13464 3/20 0.39
PRKACA P17612 2/20 0.39
MAPK8 P45983 1/20 0.38
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
PKM P14618 1/20 0.38
TACR1 P25103 1/20 0.37
F2 P00734 1/20 0.37
F10 P00742 1/20 0.37
ADRB2 P07550 1/20 0.37
ADRB1 P08588 1/20 0.37
ADRB3 P13945 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25840683 0.85 F2 (0.50) HRH3NAMPTHTTCTPS1MAPT
SCHEMBL20014224 0.84 HRH3 (0.48) HRH3NAMPTHTTCTPS1MAPT
SCHEMBL20014214 0.78 F2 (0.48) HRH3F2F10
SCHEMBL13316885 0.73 F2 (0.47) HRH3NAMPTHTTMAPTALDH1A1
SCHEMBL5476951 0.68 CCNE1 (0.63) HTTMAPTGLSALDH1A1ADRB2
SCHEMBL3604447 0.66 GSTO1 (0.42) HRH3NAMPTHTTMAPTALDH1A1
SCHEMBL24101797 0.64 ALDH1A1 (0.60) HTTCTPS1MAPTROCK1PRKACA
SCHEMBL5601202 0.64 F2 (0.47) NAMPTHTTMAPTROCK1ALDH1A1
SCHEMBL19814038 0.64 F2 (0.56) MAPTALDH1A1F2F10
SCHEMBL20640385 0.64 ACKR3 (0.47) SIGMAR1F2F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3515449-B1 QUINOLINE DERIVATIVES AS CHROMOBOX (CBX) PROTEIN INHIBITORS FOR TREATING CANCER DANA FARBER CANCER INST INC (US) 2023-07-12 EP disclosed