SCHEMBL25845703

SCHEMBL25845703

NC(=O)c1ccc2c(c1)COC(=O)N2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.48
CYP11B1 P15538 2/20 0.47
CYP11B2 P19099 2/20 0.47
TSHR P16473 1/20 0.42
SYK P43405 1/20 0.41
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
PRF1 P14222 2/20 0.39
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
GRIN2C Q14957 1/20 0.39
GRIN3A Q8TCU5 1/20 0.39
KDM1A O60341 2/20 0.38
KCNH2 Q12809 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
IP6K1 Q92551 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25184590 0.88 CYP11B1 (0.47) SIRT2CYP11B1CYP11B2SYKPDE3B
SCHEMBL4395266 0.86 CYP11B1 (0.46) SIRT2CYP11B1CYP11B2SYKPDE3B
SCHEMBL4397716 0.84 CYP11B1 (0.44) SIRT2CYP11B1CYP11B2SYKPDE3B
SCHEMBL4397712 0.78 CYP11B1 (0.44) SIRT2CYP11B1CYP11B2SYKPDE3B
SCHEMBL10916724 0.77 CYP11B1 (0.51) CYP11B1CYP11B2SYKPDE3BPDE3A
SCHEMBL3597266 0.77 LMNA (0.51) CYP11B1CYP11B2SYKPDE3BPDE3A
SCHEMBL29567045 0.76 SMYD3 (0.57) SIRT2SMYD3
SCHEMBL3190474 0.76 SMYD3 (0.57) SIRT2SMYD3
Hydrochloric Acid SCHEMBL28849276 0.74 SMYD3 (0.56) SIRT2SMYD3
SCHEMBL9375237 0.74 SIRT2 (0.61) SIRT2CYP11B1CYP11B2PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023122212-A2 SUBSTITUTED PHENYL ETHYNYL PYRIDINE CARBOXAMIDES AS POTENT INHIBITORS OF SARS VIRUS SOUTHERN RESEARCH INSTITUTE (US) 2023-06-29 WO disclosed