SCHEMBL2584833

SCHEMBL2584833

O=C(NCCc1ccccc1Cl)c1noc2c1CN(S(=O)(=O)c1cc(Cl)ccc1Cl)CC2

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.44
KMT2A Q03164 3/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 5/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
GAA P10253 2/20 0.42
RAB9A P51151 2/20 0.42
RECQL P46063 1/20 0.42
HSP90AA1 P07900 2/20 0.42
TDP1 Q9NUW8 3/20 0.40
P2RX7 Q99572 1/20 0.40
LMNA P02545 3/20 0.40
POLB P06746 2/20 0.40
TP53 P04637 2/20 0.40
MAPT P10636 2/20 0.40
ALOX15 P16050 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2588879 0.81 HSP90AA1 (0.42) NPC1KMT2AMEN1ALDH1A1SMN1; SMN2
SCHEMBL2585772 0.81 TDP1 (0.41) NPC1KMT2AMEN1ALDH1A1SMN1; SMN2
SCHEMBL4264818 0.81 ALDH1A1 (0.48) KMT2AMEN1ALDH1A1TDP1POLB
SCHEMBL2582036 0.79 GAA (0.52) NPC1KMT2AALDH1A1SMN1; SMN2GAA
SCHEMBL2586645 0.78 TP53 (0.52) KMT2AMEN1ALDH1A1SMN1; SMN2GAA
SCHEMBL2585773 0.76 OPRM1 (0.46) KMT2AMEN1ALDH1A1TDP1LMNA
SCHEMBL2588237 0.74 SMN1; SMN2 (0.47) NPC1KMT2AMEN1ALDH1A1SMN1; SMN2
SCHEMBL2587258 0.74 KMT2A (0.44) KMT2AMEN1ALDH1A1SMN1; SMN2GAA
SCHEMBL2581639 0.73 GAA (0.50) NPC1KMT2AMEN1ALDH1A1SMN1; SMN2
SCHEMBL5531260 0.73 ALDH1A1 (0.45) KMT2AMEN1ALDH1A1SMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US claimed
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US disclosed