SCHEMBL25848771

SCHEMBL25848771

CNS(=O)(=O)c1ccc(C(=O)NCc2ccc(C)cc2C2CC2)s1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
USP5 P45974 1/20 0.36
HRH1 P35367 1/20 0.33
CCR3 P51677 1/20 0.33
EPHX2 P34913 5/20 0.33
RXFP1 Q9HBX9 2/20 0.33
TP53 P04637 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MAPT P10636 1/20 0.33
HDAC1 Q13547 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2C Q14957 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
P2RX7 Q99572 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25848893 0.89 EPHX2 (0.42) EPHX2KDM4C
SCHEMBL25848772 0.85 NPC1 (0.43) EPHX2RXFP1TP53KMT2AMEN1
SCHEMBL25848767 0.84 KMT2A (0.35) RXFP1TP53KMT2AMEN1TDP1
SCHEMBL25848773 0.83 P2RX7 (0.41) EPHX2KMT2AMEN1TDP1HDAC1
SCHEMBL25848757 0.83 HDAC1 (0.44) EPHX2HDAC1HDAC6
SCHEMBL25848768 0.83 KMT2A (0.39) RXFP1TP53KMT2AMEN1TDP1
SCHEMBL25848776 0.81 EPHX2 (0.42) EPHX2HDAC1HDAC6
SCHEMBL25848766 0.81 RXFP1 (0.47) EPHX2RXFP1TP53KMT2AMAPT
SCHEMBL25848775 0.77 MEN1 (0.52) KMT2AMEN1TDP1MAPTSMN1; SMN2
SCHEMBL25848805 0.77 USP5 (0.46) USP5KMT2AMEN1TDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230219921-A1 KCNT1 INHIBITORS AND METHODS OF USE PRAXIS PRECISION MEDICINES, INC. 2023-07-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230219921-A1 KCNT1 INHIBITORS AND METHODS OF USE KCNT1, KCNT2, KCNQ2 USP5 4082/4885HRH1 1751/4885CCR3 4871/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.