SCHEMBL25857242

SCHEMBL25857242

Cc1cc(Cl)cc(C(C)CO)c1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.37
GABRA1 P14867 1/20 0.34
GABRB1 P18505 1/20 0.34
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
ADRB2 P07550 1/20 0.31
TRPA1 O75762 2/20 0.31
RAPGEF4 Q8WZA2 1/20 0.31
GRN P28799 1/20 0.30
SORT1 Q99523 1/20 0.30
SCN4A P35499 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17071834 0.87 ABCB11 (0.41) ABCB11GABRA1GABRB1PSEN1PSEN2
SCHEMBL16770774 0.87 ABCB11 (0.41) ABCB11GABRA1GABRB1PSEN1PSEN2
SCHEMBL19430514 0.83 NR3C1 (0.36) GABRA1GABRB1RAPGEF4SCN4A
SCHEMBL22169021 0.80 PSEN1 (0.32) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL13238643 0.79 TSHR (0.37) GABRA1GABRB1ADRB2RAPGEF4
SCHEMBL25852597 0.79 SLC6A4 (0.33)
SCHEMBL17025364 0.78 GABRA1 (0.37) GABRA1GABRB1RAPGEF4
SCHEMBL17025386 0.78 GABRA1 (0.37) GABRA1GABRB1RAPGEF4
SCHEMBL6124148 0.78 GABRA1 (0.39) GABRA1GABRB1ADRB2TRPA1RAPGEF4
SCHEMBL20738481 0.78 ABCB11 (0.36) ABCB11TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4212531-A1 AZAINDOLE DERIVATIVES AND THEIR USE AS ERK KINASE INHIBITORS AGV Discovery (FR) 2023-07-19 EP disclosed