SCHEMBL25857437

SCHEMBL25857437

CCOCOc1cc(C=O)ccc1-c1nnc(N)nc1C

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.40
ALDH1A1 P00352 12/20 0.39
MAPT P10636 2/20 0.33
HPGD P15428 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
FDPS P14324 1/20 0.33
KDM4E B2RXH2 2/20 0.33
RXFP1 Q9HBX9 1/20 0.33
TACR2 P21452 1/20 0.33
AGPAT2 O15120 1/20 0.32
CACNA2D1 P54289 1/20 0.32
TSHR P16473 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31314385 1.00 DHFR (0.40) DHFRALDH1A1MAPTHPGDNPSR1
SCHEMBL25857425 0.85 ALDH1A1 (0.36) DHFRALDH1A1MAPTHPGDNPSR1
SCHEMBL31496006 0.84 DHFR (0.35) DHFRALDH1A1MAPTHPGDNPSR1
SCHEMBL25858043 0.84 DHFR (0.35) DHFRALDH1A1MAPTHPGDNPSR1
SCHEMBL31314084 0.83 ALDH1A1 (0.39) DHFRALDH1A1MAPTHPGDNPSR1
SCHEMBL25859343 0.83 ALDH1A1 (0.39) DHFRALDH1A1MAPTHPGDNPSR1
SCHEMBL25862076 0.81 ALDH1A1 (0.38) DHFRALDH1A1MAPTHPGDNPSR1
SCHEMBL25857680 0.81 S1PR1 (0.36) NPSR1KDM4EAGPAT2CACNA2D1TSHR
SCHEMBL31314251 0.81 CACNA2D1 (0.33) CACNA2D1TSHR
SCHEMBL31314375 0.80 ALOX5AP (0.43) MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed