SCHEMBL25857680

SCHEMBL25857680

CCOCOc1cc(C#N)ccc1-c1nnc(N)nc1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.36
HSP90AB1 P08238 1/20 0.35
TRPV4 Q9HBA0 1/20 0.35
AGPAT2 O15120 2/20 0.34
NSD2 O96028 1/20 0.34
CYP19A1 P11511 2/20 0.33
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 2/20 0.33
PRKDC P78527 1/20 0.33
EGLN2 Q96KS0 2/20 0.33
CACNA2D1 P54289 1/20 0.33
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
GRM5 P41594 1/20 0.32
NR3C2 P08235 3/20 0.32
NR3C1 P04150 2/20 0.32
PGR P06401 2/20 0.32
AR P10275 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31314251 0.89 CACNA2D1 (0.33) CACNA2D1TSHR
SCHEMBL25859018 0.88 CACNA2D1 (0.34) CACNA2D1TSHR
SCHEMBL25859156 0.84 CHRNB2 (0.37) CACNA2D1TSHR
SCHEMBL25857437 0.81 DHFR (0.40) AGPAT2CACNA2D1TSHRSMN1; SMN2NPSR1
SCHEMBL31314385 0.81 DHFR (0.40) AGPAT2CACNA2D1TSHRSMN1; SMN2NPSR1
SCHEMBL25857483 0.81 ALOX5AP (0.43)
SCHEMBL31314375 0.81 ALOX5AP (0.43)
SCHEMBL24696097 0.76 NLRP3 (0.42) HSP90AB1NSD2EGLN2KDM4E
SCHEMBL31197264 0.75 CCNK (0.47)
SCHEMBL28934506 0.74 PDE5A (0.42) S1PR1TRPV4CYP19A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed