SCHEMBL25858155

SCHEMBL25858155

C#Cc1ccc(-c2nnc(C)c3ncccc23)c(OC)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 1/20 0.39
CASP6 P55212 1/20 0.39
G6PD P11413 1/20 0.39
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
PDE2A O00408 3/20 0.36
PDE10A Q9Y233 3/20 0.36
PDE4D Q08499 2/20 0.36
PDE3A Q14432 1/20 0.36
CACNA2D1 P54289 1/20 0.35
ATM Q13315 1/20 0.35
GAK O14976 2/20 0.35
EGFR P00533 2/20 0.35
DYRK1A Q13627 1/20 0.34
GLO1 Q04760 2/20 0.34
MAPT P10636 2/20 0.33
CCR1 P32246 1/20 0.33
CCR8 P51685 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25858132 0.87 ATM (0.37) NSD2CASP6G6PDMAOAMAOB
SCHEMBL30108705 0.72 KMT2A (0.47) NSD2CASP6G6PDPDE4DATM
SCHEMBL30108834 0.72 G6PD (0.44) NSD2CASP6G6PDATMDYRK1A
SCHEMBL25299180 0.70 KDM4E (0.38) MAOAMAOBPDE4DMAPTCCR1
SCHEMBL25856341 0.70 HSP90AA1 (0.38) MAOAMAOBPDE4DPDE3AEGFR
SCHEMBL30488502 0.70 KDM4E (0.38) MAOAMAOBPDE4DMAPTCCR1
SCHEMBL25858077 0.70 KDM4E (0.35) MAOAMAOBPDE4DMAPTKDM4E
SCHEMBL30108680 0.69 NSD2 (0.43) NSD2CASP6G6PDATMEGFR
SCHEMBL30108769 0.69 NSD2 (0.43) NSD2CASP6G6PDPDE2APDE4D
SCHEMBL30108849 0.68 G6PD (0.44) NSD2CASP6G6PDATMDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed