SCHEMBL30108680

SCHEMBL30108680

COc1cc(Br)ccc1-c1nnc(Cl)c2ncccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 1/20 0.43
CASP6 P55212 1/20 0.43
G6PD P11413 1/20 0.43
GLO1 Q04760 1/20 0.37
KDM4E B2RXH2 2/20 0.36
MAPT P10636 2/20 0.36
ATM Q13315 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
LMNA P02545 1/20 0.35
GLA P06280 1/20 0.35
DYRK1A Q13627 1/20 0.35
MC4R P32245 1/20 0.35
CCR1 P32246 1/20 0.35
CCR8 P51685 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PKM P14618 1/20 0.34
EGFR P00533 2/20 0.34
SLC40A1 Q9NP59 1/20 0.34
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30108834 0.86 G6PD (0.44) NSD2CASP6G6PDGLO1KDM4E
SCHEMBL30108769 0.85 NSD2 (0.43) NSD2CASP6G6PDKDM4EMAPT
SCHEMBL30108829 0.83 THRB (0.38) MAPTMEN1KMT2ATHRB
SCHEMBL28934827 0.82 KDM4E (0.41) KDM4EMAPTMEN1KMT2ALMNA
SCHEMBL30108726 0.82 KDM4E (0.41) KDM4EMAPTMEN1KMT2ALMNA
SCHEMBL30108849 0.77 G6PD (0.44) NSD2CASP6G6PDGLO1KDM4E
SCHEMBL30108774 0.77 MAOA (0.36) MC4RTHRB
SCHEMBL30108691 0.75 THRB (0.34) KDM4EMAPTATMMEN1KMT2A
SCHEMBL25257750 0.74 AMY1A (0.39) KDM4EMAPTATMMEN1KMT2A
SCHEMBL28934467 0.73 PRNP (0.38) MAPTMEN1KMT2ATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115433163-A NLRP3 inflammasome inhibitor and application thereof 药捷安康(南京)科技股份有限公司 2022-12-06 CN disclosed