SCHEMBL25858194

SCHEMBL25858194

CC#Cc1ccc(-c2nnc(N)c3ncccc23)c(O)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 4/20 0.37
HSP90AB1 P08238 2/20 0.37
IDO1 P14902 1/20 0.37
PSMB5 P28074 1/20 0.37
KDM4E B2RXH2 6/20 0.36
COMT P21964 1/20 0.35
SLC6A2 P23975 3/20 0.34
HTT P42858 3/20 0.34
MMP14 P50281 2/20 0.34
CYP1A2 P05177 2/20 0.33
MEN1 O00255 2/20 0.33
USP2 O75604 2/20 0.33
ALDH1A1 P00352 2/20 0.33
LMNA P02545 2/20 0.33
TP53 P04637 2/20 0.33
HPGD P15428 2/20 0.33
ALOX15 P16050 2/20 0.33
MAPK1 P28482 2/20 0.33
KMT2A Q03164 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25856341 0.85 HSP90AA1 (0.38) HSP90AA1HSP90AB1IDO1PSMB5KDM4E
SCHEMBL25858206 0.84 KDM4E (0.34) IDO1KDM4ECOMTSLC6A2HTT
SCHEMBL25856433 0.84 KDM4E (0.41) KDM4ECYP1A2MEN1KMT2ACYP1A1
SCHEMBL27355944 0.78 HSP90AA1 (0.38) HSP90AA1HSP90AB1IDO1PSMB5KDM4E
SCHEMBL24855472 0.76 KDM4E (0.42) HSP90AA1HSP90AB1IDO1PSMB5KDM4E
SCHEMBL25858838 0.72 ALDH1A1 (0.45) CYP1A2ALDH1A1LMNATP53CYP1A1
SCHEMBL25861298 0.71 KDM4E (0.41) KDM4E
SCHEMBL30488502 0.71 KDM4E (0.38) HSP90AA1HSP90AB1IDO1PSMB5KDM4E
SCHEMBL25299180 0.71 KDM4E (0.38) HSP90AA1HSP90AB1IDO1PSMB5KDM4E
SCHEMBL25858493 0.71 BACE1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed