SCHEMBL25856433

SCHEMBL25856433

CC#Cc1ccc(-c2nnc(N)c3ccccc23)c(O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
CYP1A1 P04798 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP1B1 Q16678 2/20 0.40
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
NR1I2 O75469 3/20 0.32
SMARCA2 P51531 3/20 0.32
SMARCA4 P51532 3/20 0.32
PBRM1 Q86U86 3/20 0.32
BRD4 O60885 1/20 0.32
EP300 Q09472 1/20 0.31
HNF4A P41235 1/20 0.31
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30
TLR9 Q9NR96 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
ATR Q13535 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25861298 0.86 KDM4E (0.41) KDM4EESR1ESR2NR1I2SMARCA2
SCHEMBL25858194 0.84 HSP90AA1 (0.37) KDM4ECYP1A1CYP1A2CYP1B1MEN1
SCHEMBL25854476 0.83 KDM4E (0.43) KDM4EESR1ESR2NR1I2SMARCA2
SCHEMBL25858838 0.82 ALDH1A1 (0.45) CYP1A1CYP1A2CYP1B1
SCHEMBL25859255 0.78 CYP1A1 (0.33) KDM4ECYP1A1CYP1A2CYP1B1MEN1
SCHEMBL25858493 0.75 BACE1 (0.33)
SCHEMBL27352762 0.75 KDM4E (0.43) KDM4EESR1ESR2NR1I2SMARCA2
SCHEMBL25859518 0.75 NLRP3 (0.37)
SCHEMBL27355770 0.73 KDM4E (0.41) KDM4EESR1ESR2NR1I2SMARCA2
SCHEMBL25304800 0.73 NLRP3 (0.56) KDM4ECYP1A1CYP1A2CYP1B1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed