SCHEMBL25858206

SCHEMBL25858206

CC#Cc1ccc(-c2nnc(NC)c3ncccc23)c(O)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.34
COMT P21964 2/20 0.34
FTO Q9C0B1 1/20 0.33
SLC6A2 P23975 1/20 0.33
HTT P42858 1/20 0.33
PDE4D Q08499 2/20 0.32
CYP1A1 P04798 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP1B1 Q16678 1/20 0.32
IDO1 P14902 2/20 0.32
KDR P35968 1/20 0.31
NLRP3 Q96P20 1/20 0.31
ALDH1A1 P00352 2/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
ALOX15 P16050 1/20 0.31
ALOX12 P18054 1/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25858077 0.87 KDM4E (0.35) KDM4ECOMTFTOSLC6A2HTT
SCHEMBL25858838 0.84 ALDH1A1 (0.45) CYP1A1CYP1A2CYP1B1KDRNLRP3
SCHEMBL25858194 0.84 HSP90AA1 (0.37) KDM4ECOMTFTOSLC6A2HTT
SCHEMBL25856433 0.72 KDM4E (0.41) KDM4ECYP1A1CYP1A2CYP1B1KMT2A
SCHEMBL25856769 0.71 ALDH1A1 (0.46) KDRNLRP3ALDH1A1LMNAMAPT
SCHEMBL25854617 0.70 NLRP3 (0.52) KDM4ENLRP3
SCHEMBL25857850 0.69 NLRP3 (0.42) NLRP3EGLN1
SCHEMBL25299180 0.69 KDM4E (0.38) KDM4ECOMTSLC6A2HTTPDE4D
SCHEMBL30488502 0.69 KDM4E (0.38) KDM4ECOMTSLC6A2HTTPDE4D
SCHEMBL25856341 0.69 HSP90AA1 (0.38) KDM4ECOMTFTOSLC6A2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed