SCHEMBL2585920

SCHEMBL2585920

CCOC(=O)[C@H]1CCC(c2cc(F)cc(F)c2)=N1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XPO1 O14980 2/20 0.39
ALDH1A1 P00352 4/20 0.37
TDP1 Q9NUW8 1/20 0.37
RAB9A P51151 1/20 0.36
HSD17B10 Q99714 3/20 0.35
HPGD P15428 2/20 0.35
TSHR P16473 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
LMNA P02545 1/20 0.34
TRPM8 Q7Z2W7 1/20 0.34
KDM4E B2RXH2 3/20 0.34
MAPT P10636 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
GAA P10253 1/20 0.34
CHRM1 P11229 2/20 0.34
DPP4 P27487 1/20 0.34
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP4F2 P78329 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28907110 0.91 XPO1 (0.44) XPO1ALDH1A1TDP1LMNAMAPT
SCHEMBL2346544 0.88 ALDH1A1 (0.37) ALDH1A1TDP1RAB9AHSD17B10HPGD
SCHEMBL2346553 0.88 ALDH1A1 (0.37) ALDH1A1TDP1RAB9AHSD17B10HPGD
SCHEMBL28674986 0.87 HSD17B10 (0.36) ALDH1A1TDP1RAB9AHSD17B10GAA
SCHEMBL28674985 0.87 HSD17B10 (0.36) ALDH1A1TDP1RAB9AHSD17B10GAA
SCHEMBL2584512 0.87 TRPM8 (0.46) ALDH1A1TDP1RAB9AHSD17B10HPGD
SCHEMBL22040222 0.86 NR3C2 (0.43) ALDH1A1TDP1RAB9AHSD17B10HPGD
SCHEMBL2344446 0.83 ALDH1A1 (0.46) ALDH1A1TDP1TSHRLMNAKDM4E
SCHEMBL2344442 0.83 ALDH1A1 (0.46) ALDH1A1TDP1TSHRLMNAKDM4E
SCHEMBL15832431 0.83 ALDH1A1 (0.38) ALDH1A1RAB9AKDM4EMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109476639-B Pyrrolidine derivatives 橘生药品工业股份有限公司 2021-02-26 CN disclosed
US-8048878-B2 Two cyclic cinnamide compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2011-11-01 US disclosed