SCHEMBL25859435

SCHEMBL25859435

CNc1cc(C)c(-c2ccc(C=C(Br)Br)cc2O)nn1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IL1B P01584 6/20 0.40
TNF P01375 1/20 0.38
NLRP3 Q96P20 6/20 0.36
CHRM1 P11229 1/20 0.35
LRRK2 Q5S007 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25859375 0.79
SCHEMBL25859262 0.75 IL1B (0.43) IL1BTNFNLRP3CHRM1
SCHEMBL25859574 0.73 NLRP3 (0.43) IL1BTNFNLRP3CHRM1
SCHEMBL25857850 0.72 NLRP3 (0.42) IL1BTNFNLRP3CHRM1
SCHEMBL25861786 0.70 IL1B (0.39) IL1BTNFNLRP3CHRM1
SCHEMBL25859161 0.68 NLRP3 (0.46) IL1BTNFNLRP3CHRM1
SCHEMBL3752323 0.66 TP53 (0.46)
SCHEMBL25854960 0.65 IL1B (0.71) IL1BTNFNLRP3
SCHEMBL25859504 0.64
SCHEMBL13082127 0.64 LCK (0.58) LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed