SCHEMBL25860642

SCHEMBL25860642

C#Cc1ccc(-c2nnc(NCC3CCCO3)c3ccccc23)c(OCOCC)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 2/20 0.50
CACNA2D1 P54289 1/20 0.43
MAPT P10636 5/20 0.42
MAPK1 P28482 5/20 0.42
ALDH1A1 P00352 4/20 0.42
KMT2A Q03164 4/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
NPSR1 Q6W5P4 3/20 0.42
HTT P42858 3/20 0.42
BLM P54132 2/20 0.42
NPC1 O15118 2/20 0.42
GLA P06280 2/20 0.42
RECQL P46063 1/20 0.42
KDM4E B2RXH2 5/20 0.40
LMNA P02545 3/20 0.40
HSD17B10 Q99714 1/20 0.40
TP53 P04637 2/20 0.39
MEN1 O00255 2/20 0.39
HIF1A Q16665 2/20 0.39
UTS2R Q9UKP6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25860539 0.91 NLRP3 (0.49) NLRP3CACNA2D1MAPTMAPK1ALDH1A1
SCHEMBL25300749 0.86 NLRP3 (0.49) NLRP3CACNA2D1MAPTMAPK1ALDH1A1
SCHEMBL30488532 0.86 NLRP3 (0.49) NLRP3CACNA2D1MAPTMAPK1ALDH1A1
SCHEMBL30488586 0.83 NLRP3 (0.57) NLRP3MAPTMAPK1ALDH1A1KMT2A
SCHEMBL25302500 0.83 NLRP3 (0.57) NLRP3MAPTMAPK1ALDH1A1KMT2A
SCHEMBL25296656 0.83 CACNA2D1 (0.42) CACNA2D1MAPTMAPK1ALDH1A1KMT2A
SCHEMBL25256876 0.83 CACNA2D1 (0.42) CACNA2D1MAPTMAPK1ALDH1A1KMT2A
SCHEMBL25862420 0.83 CACNA2D1 (0.42) CACNA2D1MAPTMAPK1ALDH1A1KMT2A
SCHEMBL25300817 0.82 GBA1 (0.35) NLRP3MAPK1ALDH1A1KMT2AHTT
SCHEMBL25300818 0.82 GBA1 (0.35) NLRP3MAPK1ALDH1A1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed