SCHEMBL25864163

SCHEMBL25864163

C#Cc1ccc(-c2nnc(N[C@@H]3CCCN(S(=O)(=O)C4CC4)C3)c3ccccc23)c(O)c1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 11/20 0.45
ALDH1A1 P00352 2/20 0.40
IL1B P01584 3/20 0.39
KDM4E B2RXH2 2/20 0.37
HSD17B10 Q99714 1/20 0.37
GAA P10253 2/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
KAT2B Q92831 1/20 0.34
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28934545 0.91 NLRP3 (0.49) NLRP3ALDH1A1IL1BKDM4EHSD17B10
SCHEMBL28934549 0.91 NLRP3 (0.49) NLRP3ALDH1A1IL1BKDM4EHSD17B10
SCHEMBL25864158 0.91 NLRP3 (0.47) NLRP3ALDH1A1IL1B
SCHEMBL25855239 0.87 NLRP3 (0.38) NLRP3ALDH1A1IL1B
SCHEMBL25864239 0.86 NLRP3 (0.49) NLRP3IL1BCYP11B1CYP11B2
SCHEMBL25297240 0.85 NLRP3 (0.62) NLRP3IL1BKAT2B
SCHEMBL25256054 0.85 NLRP3 (0.62) NLRP3IL1BKAT2B
SCHEMBL30488518 0.85 NLRP3 (0.62) NLRP3IL1BKAT2B
SCHEMBL25854968 0.84 NLRP3 (0.47) NLRP3ALDH1A1IL1BKDM4EHSD17B10
SCHEMBL25855241 0.84 NLRP3 (0.48) NLRP3ALDH1A1IL1BKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed